SCHEMBL7698283

SCHEMBL7698283

CC(C)(C)OC(=O)NN1CCC(CCN2CCC(c3c[nH]c4ccccc34)CC2)CC1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 1/20 0.51
ADRA1D P25100 3/20 0.50
HTR2A P28223 4/20 0.49
HTR7 P34969 4/20 0.49
DRD2 P14416 3/20 0.49
KCNH2 Q12809 1/20 0.49
KDM4E B2RXH2 1/20 0.49
BRD4 O60885 1/20 0.49
ALDH1A1 P00352 1/20 0.49
POLB P06746 1/20 0.49
CREBBP Q92793 1/20 0.49
DRD4 P21917 1/20 0.49
DRD3 P35462 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6133832 0.81 CCR2 (0.66) ADRA1D
SCHEMBL11995164 0.78 ADRA1D (0.53) ADRA1DHTR2AHTR7DRD2KCNH2
SCHEMBL11995186 0.77 ADRA1D (0.56) ADRA1DHTR2AHTR7DRD2KCNH2
SCHEMBL7700873 0.76 ADRA1D (0.65) ADRA1DDRD2DRD4DRD3
SCHEMBL11995191 0.76 CYP2D6 (0.56) ADRA1DHTR2AHTR7DRD2KCNH2
SCHEMBL557776 0.75 KDM4E (0.70) CHRM4ADRA1DKDM4EBRD4ALDH1A1
Hydrochloric Acid SCHEMBL1703924 0.74 KDM4E (0.68) CHRM4ADRA1DKDM4EBRD4ALDH1A1
SCHEMBL14306777 0.74 ADRA1D (0.80) ADRA1DKDM4E
SCHEMBL27887336 0.73 HTR2A (0.52) ADRA1DHTR2AHTR7DRD2KCNH2
SCHEMBL373860 0.73 KDM4E (0.60) ADRA1DHTR2AHTR7DRD2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002079190-A1 3-SUBSTITUTED INDOLES AS CHEMOKINE ANTAGONISTS SMITHKLINE BEECHAM P.L.C. (GB) 2002-10-10 WO disclosed