SCHEMBL7698568

SCHEMBL7698568

COCCOc1cc(NC(=O)O)c([N+](=O)[O-])cc1-c1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.43
MAPT P10636 5/20 0.43
KDM4E B2RXH2 2/20 0.43
ABCB1 P08183 5/20 0.42
ABCC1 P33527 4/20 0.42
HCAR3 P49019 1/20 0.41
HTT P42858 1/20 0.41
BCL9 O00512 2/20 0.39
CTNNB1 P35222 2/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
PTGER4 P35408 1/20 0.39
RAB9A P51151 1/20 0.39
CHEK1 O14757 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7146551 0.87 ABCB1 (0.39) ALDH1A1MAPTKDM4EABCB1ABCC1
SCHEMBL7698560 0.83 DHODH (0.38) ALDH1A1MAPTABCB1ABCC1MEN1
SCHEMBL7145942 0.79 KCNQ4 (0.36) ALDH1A1MAPTKDM4EABCB1ABCC1
SCHEMBL7467490 0.76 ABCB1 (0.46) ALDH1A1MAPTABCB1ABCC1MEN1
SCHEMBL7139923 0.74 ALDH1A1 (0.40) ALDH1A1MAPTABCB1ABCC1HTT
SCHEMBL7703599 0.74 ABCB1 (0.44) ALDH1A1MAPTABCB1ABCC1HTT
SCHEMBL17728882 0.74 RAB9A (0.57) ALDH1A1MAPTHCAR3MEN1LMNA
SCHEMBL17728883 0.74 RAB9A (0.57) ALDH1A1MAPTHCAR3MEN1LMNA
SCHEMBL7138373 0.74 ABCB1 (0.47) ALDH1A1MAPTABCB1ABCC1HTT
SCHEMBL7142774 0.73 KCNQ4 (0.38) ALDH1A1MAPTABCB1ABCC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1224174-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2002-07-24 EP disclosed
WO-2001029011-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-04-26 WO disclosed