SCHEMBL7699374

SCHEMBL7699374

Fc1ccc(-c2nc3c(Br)c4ccccc4c(Br)c3nc2-c2ccc(F)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.47
MAPK14 Q16539 4/20 0.47
MAPK10 P53779 1/20 0.47
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C19 P33261 2/20 0.46
KDM4E B2RXH2 1/20 0.46
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
ALDH1A1 P00352 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
SCN9A Q15858 3/20 0.41
GPR84 Q9NQS5 1/20 0.40
BCHE P06276 1/20 0.40
CYP2C9 P11712 1/20 0.39
GRM2 Q14416 2/20 0.38
ADORA1 P30542 2/20 0.38
TNKS O95271 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7695816 0.85 ALDH1A1 (0.43) ADORA2AMAPK14CYP1A2CYP3A4CYP2C19
SCHEMBL7692593 0.84 DHFR (0.43) ADORA2AMAPK10KDM4EHPGDHTT
SCHEMBL14667006 0.82 MAPK14 (0.43) ADORA2AMAPK14MAPK10CYP1A2CYP3A4
SCHEMBL7696278 0.81 TDP1 (0.52) ADORA2AKDM4EHTTNPSR1L3MBTL1
SCHEMBL7692244 0.77 KDM4E (0.56) ADORA2ACYP1A2KDM4EHPGDHTT
SCHEMBL12131275 0.76 MAPK14 (0.44) ADORA2AMAPK14MAPK10CYP1A2CYP3A4
SCHEMBL16702152 0.73 DHFR (0.47) ADORA2ACYP1A2CYP3A4KDM4EHPGD
SCHEMBL5555772 0.72 CYP1A2 (0.56) ADORA2AMAPK14CYP1A2CYP3A4CYP2C19
SCHEMBL27139390 0.71 MAPK14 (0.53) ADORA2AMAPK14MAPK10KDM4EL3MBTL1
SCHEMBL71619 0.71 MAPK14 (0.81) ADORA2AMAPK14MAPK10KDM4ENPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002094796-A2 BENZO[G]QUINOXALINE DERIVATIVES AS EFFECTIVE COMPOUNDS AGAINST INFECTIOUS DISEASES AXXIMA PHARMACEUTICALS AG (DE) 2002-11-28 WO disclosed