SCHEMBL7699393

SCHEMBL7699393

O=S(=O)=Nc1ncccn1

nearest known ligand 0.30

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 1/20 0.30
HSP90AA1 P07900 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8354280 0.70 ADRA2A (0.47) HDAC8HSP90AA1
SCHEMBL1854476 0.67
SCHEMBL1388023 0.67
SCHEMBL1854477 0.67
SCHEMBL29919450 0.65 HDAC8 (0.39) HDAC8HSP90AA1
SCHEMBL1352941 0.65 HSP90AA1 (0.39) HDAC8HSP90AA1
SCHEMBL2469365 0.65 HDAC8 (0.39) HDAC8HSP90AA1
SCHEMBL1029555 0.63
SCHEMBL4717596 0.62
SCHEMBL3050642 0.61

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-9110840-A None JP disclosed
JP-7017972-A None JP disclosed
CN-1115339-C Novel sulfonylaminopyrimidines HOFFMANN LA ROCHE (CH) 2003-07-23 CN disclosed
CN-1115339-C Novel sulfonylaminopyrimidines HOFFMANN LA ROCHE (CH) 2003-07-23 CN disclosed
WO-2002083650-A1 NOVEL SULFONYLAMINO-PYRIMIDINES ACTELION PHARMACEUTICALS LTD (CH) 2002-10-24 WO disclosed
WO-2002083650-A1 NOVEL SULFONYLAMINO-PYRIMIDINES ACTELION PHARMACEUTICALS LTD (CH) 2002-10-24 WO disclosed
CN-1050839-C Novel sulfonylamino pyrimidines HOFFMANN LA ROCHE (CH) 2000-03-29 CN disclosed
CN-1050839-C Novel sulfonylamino pyrimidines HOFFMANN LA ROCHE (CH) 2000-03-29 CN disclosed
EP-0633259-B1 Sulfonylaminopyrimidines, their preparation and their use as medicine HOFFMANN LA ROCHE (CH) 1999-01-13 EP disclosed
EP-0633259-B1 Sulfonylaminopyrimidines, their preparation and their use as medicine HOFFMANN LA ROCHE (CH) 1999-01-13 EP disclosed
JP-H09110840-A NEW SULFONYLAMINOPYRIMIDINES F HOFFMANN LA ROCHE AG 1997-04-28 JP disclosed
US-5541186-A ENDOTHELIN RECEPTOR INHIBITORS HOFFMANN-LA ROCHE INC. (US) 1996-07-30 US disclosed
US-5541186-A ENDOTHELIN RECEPTOR INHIBITORS HOFFMANN-LA ROCHE INC. (US) 1996-07-30 US disclosed
CN-1106007-A Novel sulfonylamino pyrimidines HOFFMANN LA ROCHE (CH) 1995-08-02 CN disclosed
CN-1106007-A Novel sulfonylamino pyrimidines HOFFMANN LA ROCHE (CH) 1995-08-02 CN disclosed
JP-H0717972-A NOVEL SULFONYLAMINOPYRIMIDINE F HOFFMANN LA ROCHE AG 1995-01-20 JP disclosed
EP-0633259-A1 Sulfonylaminopyrimidines, their preparation and their use as medicine F. HOFFMANN-LA ROCHE AG (CH) 1995-01-11 EP disclosed
EP-0633259-A1 Sulfonylaminopyrimidines, their preparation and their use as medicine F. HOFFMANN-LA ROCHE AG (CH) 1995-01-11 EP disclosed
US-3716537-A CERTAIN THENOYL DERIVATIVES OF BENZENSULFONYLAMINOPYRIMIDINES BOEHRINGER MANNHEIM GMBH 1973-02-13 US disclosed
US-3711564-A NOVEL SULFONYLAMINOPYRIMIDINES AND COMPOSITIONS CONTAINING THEM BOEHRINGER MANNHEIM GMBH 1973-01-16 US disclosed