SCHEMBL7700609

SCHEMBL7700609

Cc1nc2c(C)cccn2c(=O)c1CCCN1CCC(c2coc3cc(F)ccc23)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.47
HTR1A P08908 2/20 0.47
CYP2D6 P10635 2/20 0.47
TSHR P16473 2/20 0.47
PMP22 Q01453 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
KDM4E B2RXH2 2/20 0.47
HPGD P15428 2/20 0.47
MEN1 O00255 1/20 0.47
CYP3A4 P08684 1/20 0.47
MAPT P10636 1/20 0.47
PKM P14618 1/20 0.47
THPO P40225 1/20 0.47
KMT2A Q03164 1/20 0.47
ADRA2A P08913 4/20 0.46
ADRA2B P18089 4/20 0.46
ADRA2C P18825 4/20 0.46
ADRA1A P35348 4/20 0.46
DRD2 P14416 9/20 0.45
HTR2A P28223 8/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7701569 0.86 HTR2C (0.61) HTR2CHTR1ACYP2D6TSHRPMP22
Ocaperidone SCHEMBL122321 0.82 DRD2 (0.66) HTR2CHTR1ACYP2D6TSHRPMP22
Ocaperidone SCHEMBL29710913 0.82 DRD2 (0.66) HTR2CHTR1ACYP2D6TSHRPMP22
SCHEMBL7699932 0.81 DRD2 (0.55) HTR2CHTR1ACYP2D6TSHRPMP22
Ocaperidone SCHEMBL4590337 0.78 HTR2A (0.61) HTR2CHTR1ACYP2D6TSHRPMP22
SCHEMBL7703857 0.78 DRD2 (0.51) HTR2CHTR1ACYP2D6TSHRPMP22
SCHEMBL9285766 0.77 HTR1A (0.47) HTR2CHTR1ACYP2D6TSHRPMP22
SCHEMBL7697170 0.77 DRD2 (0.53) HTR2CHTR1ACYP2D6TSHRPMP22
Ocaperidone SCHEMBL4590606 0.77 HTR2A (0.59) HTR2CHTR1ACYP2D6TSHRPMP22
Ocaperidone SCHEMBL4590272 0.76 DRD2 (0.59) HTR2CHTR1ACYP2D6TSHRPMP22

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6348457-B1 ANTAGONIZING RESERPINE IN MAMMALS JANSSEN PHARMACEUTICA N.V. (BE) 2002-02-19 US disclosed