SCHEMBL7701640

SCHEMBL7701640

O=C(CI)c1cnc(OCF)cn1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 1/20 0.39
BACE1 P56817 16/20 0.35
BACE2 Q9Y5Z0 12/20 0.35
CYP2D6 P10635 5/20 0.35
CYP2C9 P11712 1/20 0.35
KCNH2 Q12809 1/20 0.35
GRIN2B Q13224 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31379016 0.80 SIRT6 (0.46) SIRT6BACE1BACE2CYP2D6
SCHEMBL991368 0.80 SIRT6 (0.46) SIRT6BACE1BACE2CYP2D6
SCHEMBL15476644 0.79 SIRT6 (0.62) SIRT6BACE1BACE2CYP2D6CYP2C9
SCHEMBL991518 0.76 MAPK1 (0.46) SIRT6BACE1BACE2CYP2D6CYP2C9
SCHEMBL20685032 0.75 BACE1 (0.43) SIRT6BACE1BACE2CYP2D6CYP2C9
SCHEMBL23538019 0.73 POLB (0.45) SIRT6
SCHEMBL14387783 0.71 SIRT6 (0.57) SIRT6
SCHEMBL15705171 0.68 NPC1 (0.62) BACE1BACE2CYP2D6CYP2C9KCNH2
SCHEMBL2108443 0.67 SIRT6 (0.43) SIRT6BACE1BACE2
SCHEMBL15751614 0.67 SIRT6 (0.61) SIRT6BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011138293-A1 2,5,6,7-TETRAHYDRO-[1,4]OXAZEPIN-3-YLAMINE OR 2,3,6,7-TETRAHYDRO-[1,4]OXAZEPIN-5-YLAMINE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2011-11-10 WO disclosed