SCHEMBL7702065

SCHEMBL7702065

O=c1nc(-c2ccc(F)c(F)c2)c2ccccc2[nH]1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.65
HSD17B10 Q99714 2/20 0.65
ALDH1A1 P00352 2/20 0.65
HPGD P15428 1/20 0.65
TSHR P16473 1/20 0.65
KMT2A Q03164 2/20 0.52
MEN1 O00255 1/20 0.52
CASP1 P29466 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
PDE3B Q13370 1/20 0.47
PDE3A Q14432 1/20 0.47
IDO1 P14902 1/20 0.43
CTSV O60911 1/20 0.42
CTSL P07711 1/20 0.42
TRPA1 O75762 1/20 0.42
APP P05067 2/20 0.40
MAOB P27338 1/20 0.40
CYP1A1 P04798 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP1B1 Q16678 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8621648 0.84 KDM4E (0.89) KDM4EHSD17B10ALDH1A1HPGDTSHR
SCHEMBL6329236 0.83 KDM4E (0.76) KDM4EHSD17B10ALDH1A1HPGDTSHR
SCHEMBL4094165 0.80 KDM4E (0.76) KDM4EHSD17B10ALDH1A1HPGDTSHR
SCHEMBL17367227 0.80 KDM4E (0.93) KDM4EHSD17B10ALDH1A1HPGDTSHR
SCHEMBL4142958 0.79 KDM4E (1.00) KDM4EHSD17B10ALDH1A1HPGDTSHR
Lithium SCHEMBL30669498 0.78 KDM4E (0.96) KDM4EHSD17B10ALDH1A1HPGDTSHR
SCHEMBL6329154 0.77 ALDH1A1 (0.61) KDM4EHSD17B10ALDH1A1HPGDTSHR
SCHEMBL28022669 0.75 HSD17B10 (0.78) KDM4EHSD17B10ALDH1A1HPGDTSHR
SCHEMBL29130443 0.75 KDM4E (0.71) KDM4EHSD17B10ALDH1A1HPGDTSHR
SCHEMBL29130442 0.73 HPGD (0.64) KDM4EHSD17B10ALDH1A1HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6358959-B1 FOR THERAPY OF BENIGN PROSTATIC HYPERPLASIA MERCK & CO., INC. 2002-03-19 US disclosed
WO-2000043374-A1 POLYAZANAPHTHALENONE DERIVATIVES USEFUL AS ALPHA 1A ADRENOCEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2000-07-27 WO disclosed