SCHEMBL7702223

SCHEMBL7702223

C=CC(CCC(=O)O)CC(=O)O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.54
SLC6A4 P31645 1/20 0.54
BLM P54132 1/20 0.54
SLC6A3 Q01959 1/20 0.54
MEN1 O00255 1/20 0.54
CYP2D6 P10635 1/20 0.54
TSHR P16473 1/20 0.54
NFKB1 P19838 1/20 0.54
CYP2C19 P33261 1/20 0.54
KMT2A Q03164 1/20 0.54
FOLH1 Q04609 4/20 0.46
TET2 Q6N021 3/20 0.39
KDM4A O75164 2/20 0.39
KDM4C Q9H3R0 2/20 0.39
KDM2A Q9Y2K7 2/20 0.39
TET3 O43151 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11528893 0.88 CYP2D6 (0.60) SLC6A2SLC6A4BLMSLC6A3MEN1
SCHEMBL27906416 0.85 HDAC3 (0.46) SLC6A2SLC6A4BLMSLC6A3MEN1
SCHEMBL7707787 0.84 SLC6A2 (0.41) SLC6A2SLC6A4BLMSLC6A3MEN1
SCHEMBL4280331 0.83 SLC22A6 (0.43) SLC6A2SLC6A4BLMSLC6A3MEN1
SCHEMBL29237760 0.82 SLC6A2 (0.39) SLC6A2SLC6A4BLMSLC6A3MEN1
SCHEMBL7705158 0.80 TSHR (0.52) SLC6A2SLC6A4BLMSLC6A3MEN1
SCHEMBL8006389 0.80 GPR84 (0.39) SLC6A2SLC6A4BLMSLC6A3MEN1
SCHEMBL27375200 0.80 CYP2D6 (0.52) SLC6A2SLC6A4BLMSLC6A3MEN1
SCHEMBL27801322 0.79 SLC6A2 (0.42) SLC6A2SLC6A4BLMSLC6A3MEN1
SCHEMBL27906400 0.78 TSHR (0.42) SLC6A2SLC6A4BLMSLC6A3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170260190-A1 SUBSTITUTED PYRIMIDINE COMPOUNDS AND METHODS OF USE AND MANUFACTURE DUQUESNE UNIVERSITY OF THE HOLY SPIRIT (US) 2017-09-14 US disclosed
US-20170260190-A1 SUBSTITUTED PYRIMIDINE COMPOUNDS AND METHODS OF USE AND MANUFACTURE DUQUESNE UNIVERSITY OF THE HOLY SPIRIT (US) 2017-09-14 US disclosed
US-9650384-B2 Substituted pyrimidine compounds and methods of use and manufacture DUQUESNE UNIVERSITY OF THE HOLY GHOST (US) 2017-05-16 US disclosed
US-9650384-B2 Substituted pyrimidine compounds and methods of use and manufacture DUQUESNE UNIVERSITY OF THE HOLY GHOST (US) 2017-05-16 US disclosed
WO-2016022881-A1 SUBSTITUTED PYRIMIDINE COMPOUNDS AND METHODS OF USE AND MANUFACTURE DUQUESNE UNIVERSITY OF THE HOLY SPIRIT (US) 2016-02-11 WO disclosed
US-20160039830-A1 Substituted Pyrimidine Compounds and Methods of Use and Manufacture DUQUESNE UNIVERSITY OF THE HOLY SPIRIT 2016-02-11 US disclosed
US-20160039830-A1 Substituted Pyrimidine Compounds and Methods of Use and Manufacture DUQUESNE UNIVERSITY OF THE HOLY SPIRIT 2016-02-11 US disclosed
US-8946468-B2 Process for producing ester compound having an internal unsaturated bond or cyclic olefin JX NIPPON OIL & ENERGY CORPORATION (JP) 2015-02-03 US disclosed
US-20120316360-A1 PROCESS FOR PRODUCING ESTER COMPOUND HAVING a,ß-UNSATURATED BOND OSAKA UNIVERSITY (JP) 2012-12-13 US disclosed
US-6348623-B2 (CO)POLYMERS OF 1-ACETOXY-2-METHOXY-3-BUTENE FOR EXAMPLE; CAN COPOLYMERIZE WITH VINYL ACETATE; REACTING ACETOACETOXY FUNCTIONAL POLYMER WITH AMMONIA OR PRIMARY OR SECONDARY AMINES TO FORM ENAMINE FUNCTIONAL POLYMERS; COATINGS EASTMAN CHEMICAL COMPANY 2002-02-19 US disclosed
US-20010051690-A1 Polymers of 3-butene esters, their preparation and use EASTMAN CHEMICAL COMPANY 2001-12-13 US disclosed
US-6228949-B1 ACETOACETOXY-DERIVATIZED HOMO OR CO-POLY(3,4-EPOXY-1-BUTENE) WHEREBY THE ACETOACETOXY GROUPS HAVE BEEN REACTED WITH AMMONIA, PRIMARY OR SECONDARY AMINE TO FORM ENAMINE FUNCTIONAL GROUPS; HIGH MOLECULAR WEIGHT COATINGS, ADHESIVES EASTMAN CHEMICAL COMPANY 2001-05-08 US disclosed
US-6160057-A Polymers of 3-butene esters, their preparation and use EASTMAN CHEMICAL COMPANY (US) 2000-12-12 US disclosed
US-6121400-A FREE-RADICAL POLYMERIZATION PRODUCT; FOR COATING COMPOSITIONS SUCH AS INKS, ADHESIVES, PAINTS, AND FILMS EASTMAN CHEMICAL COMPANY (US) 2000-09-19 US disclosed
US-6121399-A Polymers of 3-butene esters, their preparation and use EASTMAN CHEMICAL COMPANY (US) 2000-09-19 US disclosed
EP-1023340-A1 POLYMERS OF 3-BUTENE ESTERS, THEIR PREPARATION AND USE EASTMAN CHEMICAL COMPANY (US) 2000-08-02 EP disclosed
WO-1999020666-A1 POLYMERS OF 3-BUTENE ESTERS, THEIR PREPARATION AND USE EASTMAN CHEMICAL COMPANY (US) 1999-04-29 WO disclosed
US-4734100-A Process for printing or dyeing cellulose-containing textile material CIBA-GEIGY CORPORATION (US) 1988-03-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170260190-A1 SUBSTITUTED PYRIMIDINE COMPOUNDS AND METHODS OF USE AND MANUFACTURE DHFR, FOLR1, DPYD SLC6A2 2626/4885SLC6A4 1046/4885BLM 2645/4885
US-20120316360-A1 PROCESS FOR PRODUCING ESTER COMPOUND HAVING a,ß-UNSATURATED BOND COASY, OXER1, ACSL1 SLC6A2 4763/4885SLC6A4 4832/4885BLM 4594/4885
US-20010051690-A1 Polymers of 3-butene esters, their preparation and use CCNT1, C1S, H1-3 SLC6A2 3999/4885SLC6A4 4554/4885BLM 3723/4885
US-20160039830-A1 Substituted Pyrimidine Compounds and Methods of Use and Manufacture DHFR, FOLR1, DPYD SLC6A2 2626/4885SLC6A4 1046/4885BLM 2645/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.