SCHEMBL770258

SCHEMBL770258

O=C(NCCC(=O)N1CCCC2CCCCC21)c1cccc2ccccc12

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PREP P48147 8/20 0.57
FAP Q12884 2/20 0.57
DPP8 Q6V1X1 1/20 0.57
DPP9 Q86TI2 1/20 0.57
HPGD P15428 1/20 0.48
BCHE P06276 1/20 0.48
TGM2 P21980 1/20 0.45
DRD4 P21917 2/20 0.45
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
DPP7 Q9UHL4 2/20 0.44
CNR1 P21554 3/20 0.44
CNR2 P34972 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
PPARG P37231 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL771667 0.94 PREP (0.55) PREPFAPDPP8DPP9HPGD
SCHEMBL772132 0.88 PREP (0.60) PREPFAPDPP8DPP9LMNA
SCHEMBL770007 0.83 PREP (0.60) PREPFAPDPP7
SCHEMBL770966 0.83 RAB9A (0.51) PREPFAPDPP8DPP9DPP7
SCHEMBL770891 0.82 KMT2A (0.49) PREPFAPDPP8DPP9HPGD
SCHEMBL770799 0.82 DPP4 (0.60) PREPFAPDPP7NPC1RAB9A
SCHEMBL769774 0.79 SLC6A4 (0.51) HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL770920 0.78 RAB9A (0.54) HPGDPOLBNPC1RAB9ASMN1; SMN2
SCHEMBL770599 0.78 DRD3 (0.48)
SCHEMBL770850 0.77 HDAC1 (0.51) POLBCNR2NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130303522-A1 INHIBITOR COMPOUNDS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 LABORATORIOS SALVAT, S.A. (ES) 2013-11-14 US disclosed
US-20120071466-A1 INHIBITOR COMPOUNDS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 LABORATORIOS SALVAT, S.A. (ES) 2012-03-22 US disclosed
US-20120071466-A1 INHIBITOR COMPOUNDS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 LABORATORIOS SALVAT, S.A. (ES) 2012-03-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130303522-A1 INHIBITOR COMPOUNDS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 HSD11B1, HSD17B1, HSD11B2 PREP 900/4885FAP 2352/4885DPP8 1886/4885
US-20120071466-A1 INHIBITOR COMPOUNDS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 HSD11B1, HSD17B1, HSD11B2 PREP 907/4885FAP 2369/4885DPP8 1905/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.