SCHEMBL7702988

SCHEMBL7702988

CC(C)(C)OC(=O)C(Cn1cnc2c(N3CCC(C(=O)NC4=NCCCN4)CC3)ncnc21)NC(=O)OCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 19/20 0.44
ITGAV P06756 18/20 0.44
ITGA2B P08514 5/20 0.44
ITGB5 P18084 1/20 0.38
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4644035 1.00 ITGB3 (0.44) ITGB3ITGAVITGA2BITGB5MAPT
SCHEMBL4640251 0.92 ITGB3 (0.49) ITGB3ITGAVITGA2BITGB5
SCHEMBL4641013 0.90 ITGB3 (0.34) ITGB3ITGAVITGA2BMAPT
SCHEMBL6882095 0.88 STS (0.41) ITGB3ITGAVITGA2BMAPT
Benzene SCHEMBL6882109 0.87 MAPT (0.35) ITGB3ITGAVITGA2BMAPT
SCHEMBL6810562 0.87 ITGB3 (0.41) ITGB3ITGAVITGA2BMAPT
SCHEMBL6805791 0.86 ITGB3 (0.44) ITGB3ITGAVITGA2BMAPT
SCHEMBL27524220 0.86 ITGB3 (0.46) ITGB3ITGAVITGA2BITGB5
SCHEMBL4640164 0.86 ITGB3 (0.46) ITGB3ITGAVITGA2BITGB5
SCHEMBL6876023 0.85 SIRT2 (0.36) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1196416-A1 SUBSTITUTED PURINE DERIVATIVES AS INHIBITORS OF CELL ADHESION Aventis Pharma Deutschland GmbH (DE) 2002-04-17 EP disclosed
WO-2001002399-A1 SUBSTITUTED PURINE DERIVATIVES AS INHIBITORS OF CELL ADHESION AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-01-11 WO disclosed