SCHEMBL4640164

SCHEMBL4640164

CC(C)(C)OC(=O)[C@H](Cn1cnc2c(N3CCC(C(=O)O)CC3)ncnc21)NC(=O)OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 14/20 0.46
ITGAV P06756 14/20 0.46
CNR1 P21554 1/20 0.42
CNR2 P34972 1/20 0.42
ITGA2B P08514 1/20 0.41
ITGB5 P18084 1/20 0.41
HRH4 Q9H3N8 1/20 0.41
ADORA3 P0DMS8 1/20 0.39
ADORA2A P29274 1/20 0.39
ADORA2B P29275 1/20 0.39
ADORA1 P30542 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27524220 1.00 ITGB3 (0.46) ITGB3ITGAVCNR1CNR2ITGA2B
SCHEMBL4640844 0.91 ITGB3 (0.48) ITGB3ITGAVITGA2BITGB5HRH4
SCHEMBL6811091 0.90 ITGB3 (0.53) ITGB3ITGAVCNR1CNR2ITGA2B
SCHEMBL4640097 0.89 TDP1 (0.36) ITGB3ITGAVCNR1CNR2HRH4
SCHEMBL7702988 0.86 ITGB3 (0.44) ITGB3ITGAVITGA2BITGB5
SCHEMBL4644035 0.86 ITGB3 (0.44) ITGB3ITGAVITGA2BITGB5
SCHEMBL6810270 0.84 NPEPPS (0.34) ITGB3ITGAVCNR1CNR2HRH4
SCHEMBL6016455 0.83 HDAC6 (0.43) ITGB3ITGAV
SCHEMBL6016459 0.83 HDAC6 (0.43) ITGB3ITGAV
SCHEMBL6805979 0.83 CNR1 (0.41) ITGB3ITGAVCNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853084-B1 Substituted purine derivatives as vitronectin receptor antagonists HOECHST AG (DE) 2008-08-13 EP disclosed
US-6747016-B1 TREATING OSTEOPOROSIS IN WARM-BLOODED ANIMALS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2004-06-08 US disclosed
US-6723727-B1 VITRONECTIN RECEPTOR ANTAGONISTS; INHIBITORS OF BONE RESORPTION; OSTEOPOROSIS HOECHST AKTIENGESELLSCHAFT (DE) 2004-04-20 US disclosed
EP-1196416-B1 SUBSTITUTED PURINE DERIVATIVES AS INHIBITORS OF CELL ADHESION AVENTIS PHARMA GMBH (DE) 2004-03-24 EP disclosed
EP-1196416-A1 SUBSTITUTED PURINE DERIVATIVES AS INHIBITORS OF CELL ADHESION Aventis Pharma Deutschland GmbH (DE) 2002-04-17 EP disclosed
WO-2001002399-A1 SUBSTITUTED PURINE DERIVATIVES AS INHIBITORS OF CELL ADHESION AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-01-11 WO disclosed
EP-1065208-A1 Substituted purine derivatives as inhibitors of cell adhesion Aventis Pharma Deutschland GmbH (DE) 2001-01-03 EP disclosed
EP-0853084-A2 Substituted purine derivatives as vitronectin receptor antagonists HOECHST AKTIENGESELLSCHAFT (DE) 1998-07-15 EP disclosed