SCHEMBL7703218

SCHEMBL7703218

Nc1cc(-c2ccc(F)c(Cl)c2)cc2nc(-c3ccno3)nn12

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.37
KCNH2 Q12809 1/20 0.34
ADORA2A P29274 9/20 0.33
ADORA1 P30542 1/20 0.33
EPHB4 P54760 1/20 0.32
NISCH Q9Y2I1 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
KMO O15229 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7708813 0.91 NPC1 (0.37) NOTUMADORA2AKDM4EMEN1ALDH1A1
SCHEMBL7705951 0.85 BACE1 (0.40) NOTUMADORA2AADORA1ALDH1A1
SCHEMBL7711697 0.85 ADORA2A (0.35) ADORA2AKDM4EMEN1ALDH1A1LMNA
SCHEMBL7702990 0.83 ADORA2A (0.50) ADORA2A
SCHEMBL7711711 0.82 ALDH1A1 (0.44) ADORA2AKDM4EALDH1A1TP53
SCHEMBL7703193 0.81 ADORA2A (0.46) ADORA2AADORA1KDM4EMEN1ALDH1A1
SCHEMBL7709236 0.81 ALDH1A1 (0.48) ADORA2AKDM4EMEN1ALDH1A1LMNA
SCHEMBL7708391 0.81 ADORA2A (0.45) ADORA2AKDM4EMEN1ALDH1A1MAPT
SCHEMBL7703234 0.81 ADORA2A (0.38) ADORA2AMEN1ALDH1A1
SCHEMBL7708387 0.80 BACE1 (0.40) ADORA2AMEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed