SCHEMBL7708387

SCHEMBL7708387

Nc1cc(-c2ccccc2F)cc2nc(-c3ccno3)nn12

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.40
ADORA2A P29274 8/20 0.37
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
NFKB1 P19838 2/20 0.34
NFKB2 Q00653 2/20 0.34
RELA Q04206 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
PKM P14618 2/20 0.34
KMT2A Q03164 2/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
MEN1 O00255 1/20 0.34
MAPK1 P28482 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7708391 0.85 ADORA2A (0.45) ADORA2ANPC1RAB9ANFKB1NFKB2
SCHEMBL7487756 0.84 ADORA2A (0.56) ADORA2A
SCHEMBL7711697 0.82 ADORA2A (0.35) ADORA2ANPC1RAB9ASMN1; SMN2KMT2A
SCHEMBL7709007 0.82 ADORA2A (0.53) BACE1ADORA2ANPC1RAB9ANFKB1
SCHEMBL7711711 0.81 ALDH1A1 (0.44) ADORA2ANPC1RAB9ANFKB1NFKB2
SCHEMBL7703234 0.80 ADORA2A (0.38) ADORA2ANPC1RAB9ANFKB1NFKB2
SCHEMBL7708534 0.80 ADORA2A (0.53) BACE1ADORA2ANPC1RAB9AALDH1A1
SCHEMBL7703218 0.80 NOTUM (0.37) ADORA2AKMT2AALDH1A1MEN1
SCHEMBL7709236 0.79 ALDH1A1 (0.48) ADORA2ANPC1RAB9ANFKB1NFKB2
SCHEMBL7705951 0.78 BACE1 (0.40) BACE1ADORA2ANPC1RAB9ANFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed