SCHEMBL7704658

SCHEMBL7704658

FC(F)(F)c1c[c]cc(C(F)(F)F)c1-c1cccs1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
KDM4E B2RXH2 8/20 0.39
ALDH1A1 P00352 6/20 0.39
L3MBTL1 Q9Y468 4/20 0.39
TDP1 Q9NUW8 3/20 0.39
GAA P10253 2/20 0.39
MAPK1 P28482 2/20 0.39
RXFP1 Q9HBX9 2/20 0.37
CCNE2 O96020 1/20 0.37
CCNE1 P24864 1/20 0.37
CDK2 P24941 1/20 0.37
MAPT P10636 3/20 0.36
ACHE P22303 2/20 0.35
POLB P06746 2/20 0.35
ALOX15 P16050 1/20 0.35
HSD17B10 Q99714 1/20 0.35
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7135870 0.70 MAPT (0.52) KDM4EALDH1A1L3MBTL1TDP1MAPT
SCHEMBL10921471 0.69 ALDH1A1 (0.49) ERN1SMN1; SMN2ALDH1A1GAAACHE
SCHEMBL7465724 0.68 KIF11 (0.41) KDM4EALDH1A1L3MBTL1TDP1GAA
SCHEMBL7704656 0.68 ERN1 (0.39) ERN1SMN1; SMN2KDM4EALDH1A1L3MBTL1
SCHEMBL2752571 0.68 PDK2 (0.34) ALDH1A1HPGD
SCHEMBL732915 0.68 RPS6KB2 (0.49) ERN1SMN1; SMN2KDM4EALDH1A1GAA
SCHEMBL7702104 0.68 CYP2A6 (0.38) CCNE2CCNE1CDK2KCNH2
SCHEMBL7704882 0.67 KDM4E (0.37) KDM4EALDH1A1GAAMAPTACHE
SCHEMBL6744117 0.66 MAPT (0.44) KDM4EALDH1A1L3MBTL1TDP1MAPT
SCHEMBL5541483 0.66 L3MBTL1 (0.40) SMN1; SMN2KDM4EALDH1A1L3MBTL1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242399-A1 $g(a)-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB S.A. (BE) 2002-09-25 EP disclosed
WO-2001046167-A1 α-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB, S.A. (BE) 2001-06-28 WO disclosed