SCHEMBL7704750

SCHEMBL7704750

COC(=O)Cn1cncc1C(C)(O)c1ccc(C#N)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 3/20 0.39
AR P10275 1/20 0.39
CACNA1H O95180 4/20 0.39
POLB P06746 1/20 0.39
CYP11B1 P15538 5/20 0.37
CYP11B2 P19099 5/20 0.37
CYP3A4 P08684 2/20 0.37
CYP17A1 P05093 1/20 0.37
FNTA P49354 1/20 0.36
FNTB P49356 1/20 0.36
PGGT1B P53609 1/20 0.36
KDM4E B2RXH2 1/20 0.35
CYP1A2 P05177 1/20 0.35
GLA P06280 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
SLC22A12 Q96S37 1/20 0.35
S1PR1 P21453 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7710770 0.89 AR (0.39) S1PR3ARCACNA1HCYP11B1CYP11B2
SCHEMBL7672909 0.78 CYP17A1 (0.48) CYP11B1CYP11B2CYP3A4CYP17A1FNTA
SCHEMBL7717657 0.76 TRPA1 (0.41) S1PR3ARCACNA1HSLC22A12S1PR1
SCHEMBL7707858 0.74 HIF1A (0.36) CACNA1HPOLBFNTAFNTBPGGT1B
SCHEMBL7704743 0.70 CYP11B1 (0.55) CACNA1HCYP11B1CYP11B2FNTAFNTB
SCHEMBL7736904 0.69 S1PR3 (0.42) S1PR3CACNA1HCYP11B1CYP11B2CYP3A4
SCHEMBL7713236 0.69 CYP11B1 (0.70) CACNA1HCYP11B1CYP11B2FNTAFNTB
Hydrochloric Acid SCHEMBL7220321 0.68 FNTA (0.41) S1PR3CACNA1HCYP3A4CYP17A1FNTA
SCHEMBL5359320 0.68 CNR1 (0.45) S1PR3ARCACNA1HCYP11B1CYP11B2
SCHEMBL7673750 0.68 FNTA (0.44) S1PR3CYP11B1CYP11B2CYP3A4CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441017-B1 Inhibitors of prenyl-protein transferase MERCK & CO., INC. 2002-08-27 US disclosed
US-6358985-B1 ANTICANCER AGENT MERCK & CO., INC. 2002-03-19 US disclosed