SCHEMBL7705060

SCHEMBL7705060

CC1Oc2ccc(CN(Cc3ccc(S(N)(=O)=O)cc3)C(=O)OC(C)(C)C)cc2NC1=S

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA2 P00918 15/20 0.35
CA1 P00915 13/20 0.35
CA9 Q16790 10/20 0.35
CA12 O43570 10/20 0.35
CA4 P22748 7/20 0.35
CA14 Q9ULX7 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
NCOR2 Q9Y618 1/20 0.33
CA7 P43166 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
PARP1 P09874 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7711220 0.92 HDAC3 (0.34) HDAC3HDAC1HDAC2NCOR2PARP1
SCHEMBL7704945 0.88 HDAC3 (0.44) HDAC3HDAC1HDAC2NCOR2PARP1
SCHEMBL7704907 0.88 HSD17B10 (0.38) HDAC3HDAC1HDAC2NCOR2PARP1
SCHEMBL7704932 0.87 HDAC3 (0.35) HDAC3HDAC1HDAC2NCOR2PARP1
SCHEMBL7708363 0.86 TP53 (0.35) HDAC3HDAC1HDAC2NCOR2PARP1
SCHEMBL7711422 0.86 HSD17B10 (0.36) HDAC3HDAC1HDAC2NCOR2PARP1
SCHEMBL6309617 0.86 HDAC1 (0.43) HDAC3HDAC1HDAC2NCOR2PARP1
SCHEMBL7710786 0.86 NR1D1 (0.39) HDAC3HDAC1HDAC2NCOR2
SCHEMBL6302990 0.84 PARP1 (0.38) HDAC3HDAC1HDAC2NCOR2TDP1
SCHEMBL7711323 0.84 ALDH1A1 (0.41) TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed