SCHEMBL7705075

SCHEMBL7705075

O=c1[c]cc2c(ccc3ccccc32)o1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.46
ALDH1A1 P00352 7/20 0.46
GLA P06280 3/20 0.46
HPGD P15428 3/20 0.46
GAA P10253 3/20 0.46
TDP1 Q9NUW8 3/20 0.46
MAPT P10636 3/20 0.46
TSHR P16473 3/20 0.46
HSD17B10 Q99714 3/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
HTT P42858 1/20 0.46
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA9 Q16790 1/20 0.45
GPR55 Q9Y2T6 1/20 0.45
MAOB P27338 1/20 0.45
HNF4A P41235 1/20 0.45
MCL1 Q07820 1/20 0.45
CYP2A6 P11509 1/20 0.43
PAX8 Q06710 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25909 0.75 CA12 (0.48) KDM4EALDH1A1GLAHPGDGAA
SCHEMBL3362663 0.72 TDP1 (0.61) KDM4EALDH1A1GLAHPGDGAA
SCHEMBL30450770 0.72 TDP1 (0.61) KDM4EALDH1A1GLAHPGDGAA
SCHEMBL30588914 0.72 TDP1 (0.61) KDM4EALDH1A1GLAHPGDGAA
SCHEMBL5672210 0.70 TDP1 (0.59) KDM4EALDH1A1GLAHPGDGAA
SCHEMBL31035850 0.70 TDP1 (0.59) KDM4EALDH1A1GLAHPGDGAA
SCHEMBL2518542 0.69 ALDH1A1 (0.50) KDM4EALDH1A1GLAHPGDGAA
SCHEMBL7912365 0.67 ABCG2 (0.60) KDM4EALDH1A1GLAHPGDGAA
SCHEMBL21019890 0.67 TDP1 (0.61) KDM4EALDH1A1GLAHPGDGAA
SCHEMBL14231901 0.67 NISCH (0.59) KDM4EALDH1A1GLAHPGDGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE37556-E1 (ALKOXYPHENYL)THIAZOLE DERIVATIVES OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2002-02-19 US claimed
EP-1130017-A2 Azole derivatives and their use as superoxide radical inhibitors OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2001-09-05 EP claimed
EP-0934937-A1 Azole derivatives as superoxide radical inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1999-08-11 EP claimed
US-5643932-A PREVENTS CELL DAMAGE AFTER ISCHEMIA AND RE-PERFUSION, SUBSTITUTED THIAZOLES OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-07-01 US claimed