SCHEMBL7705183

SCHEMBL7705183

CCOC(=O)N1CCN([C@@H](C)c2ccccc2O)CC1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 6/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
CHRM2 P08172 1/20 0.58
CHRM1 P11229 1/20 0.58
TSHR P16473 2/20 0.52
LMNA P02545 3/20 0.52
ALDH1A1 P00352 7/20 0.49
PKM P14618 1/20 0.49
POLB P06746 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
MAPT P10636 3/20 0.49
L3MBTL1 Q9Y468 1/20 0.48
KDM4E B2RXH2 4/20 0.48
KMT2A Q03164 1/20 0.47
HPGD P15428 1/20 0.47
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3976528 0.76 GABRA1 (0.50) GAATSHRLMNAALDH1A1POLB
SCHEMBL5447670 0.75 ALDH1A1 (0.52) GAASMN1; SMN2CHRM2CHRM1TSHR
SCHEMBL9322403 0.75 CHRM2 (0.49) GAACHRM2CHRM1TSHRLMNA
SCHEMBL7224481 0.74 GAA (1.00) GAASMN1; SMN2TSHRLMNAALDH1A1
SCHEMBL7704915 0.73 TACR1 (0.61) SMN1; SMN2CHRM2CHRM1LMNAALDH1A1
SCHEMBL681679 0.72 ALDH1A1 (0.56) GAASMN1; SMN2CHRM2CHRM1TSHR
SCHEMBL31074064 0.71 TSHR (0.53) GAASMN1; SMN2TSHRLMNAALDH1A1
SCHEMBL10858287 0.71 TSHR (0.53) GAASMN1; SMN2TSHRLMNAALDH1A1
SCHEMBL6479504 0.71 TSHR (0.64) GAASMN1; SMN2CHRM2CHRM1TSHR
SCHEMBL6479978 0.71 TSHR (0.64) GAASMN1; SMN2CHRM2CHRM1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242399-A1 $g(a)-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB S.A. (BE) 2002-09-25 EP disclosed
WO-2001046167-A1 α-ARYLETHYLPIPERAZINE DERIVATIVES AS NEUROKININ ANTAGONISTS UCB, S.A. (BE) 2001-06-28 WO disclosed