SCHEMBL7705451

SCHEMBL7705451

NC(=O)c1cc(N2CCCC2)cc2nc(N3CCCNCC3)[nH]c12

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 6/20 0.48
CHRNA4 P43681 6/20 0.48
PIM1 P11309 1/20 0.43
CHRNA1 P02708 1/20 0.39
CHRNA7 P36544 1/20 0.39
ITGB3 P05106 3/20 0.38
ITGA2B P08514 3/20 0.38
HTR3A P46098 1/20 0.38
JAK2 O60674 1/20 0.37
HRH4 Q9H3N8 1/20 0.37
MGLL Q99685 1/20 0.37
PRKD3 O94806 1/20 0.37
PRKD1 Q15139 1/20 0.37
PRKD2 Q9BZL6 1/20 0.37
SCN9A Q15858 1/20 0.36
CASP1 P29466 1/20 0.35
CASP4 P49662 1/20 0.35
CASP5 P51878 1/20 0.35
NAMPT P43490 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5621943 0.98 CHRNB2 (0.44) CHRNB2CHRNA4PIM1ITGB3ITGA2B
SCHEMBL5620177 0.87 CHRNB2 (0.44) CHRNB2CHRNA4PIM1ITGB3ITGA2B
SCHEMBL5621961 0.86 CHRNB2 (0.43) CHRNB2CHRNA4PIM1CHRNA1CHRNA7
SCHEMBL5620211 0.84 CHRNB2 (0.41) CHRNB2CHRNA4PIM1ITGB3ITGA2B
SCHEMBL5622573 0.82 HTR3A (0.42) CHRNB2CHRNA4PIM1ITGB3ITGA2B
SCHEMBL5620821 0.82 PARP1 (0.50) CHRNB2CHRNA4
SCHEMBL5621910 0.81 HTR3A (0.48) CHRNB2CHRNA4PIM1ITGB3ITGA2B
SCHEMBL5621369 0.81 CHRM2 (0.41) CHRNB2CHRNA4PIM1ITGB3ITGA2B
SCHEMBL5621940 0.79 PARP1 (0.52) CHRNB2CHRNA4
SCHEMBL5621393 0.79 PARP1 (0.46) CHRNB2CHRNA4JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448271-B1 SUCH AS 2-(PIPERIDIN-4-YL)BENZIMIDAZOLE-4-CARBOXAMIDE; INHIBITORS OF ENZYME POLY(ADP-RIBOSE)POLYMERASE; IMPROVED WATER SOLUBILITY BASF AKTIENGESELLSCHAFT (DE) 2002-09-10 US disclosed