SCHEMBL5620177

SCHEMBL5620177

NC(=O)c1cc(N)cc2nc(N3CCCNCC3)[nH]c12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.44
CHRNA4 P43681 2/20 0.44
PIM1 P11309 2/20 0.43
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
THRB P10828 1/20 0.39
ALOX15 P16050 1/20 0.39
GFER P55789 1/20 0.39
YWHAG P61981 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HTR3A P46098 1/20 0.39
HRH4 Q9H3N8 1/20 0.38
NAMPT P43490 1/20 0.38
HTT P42858 1/20 0.38
IKBKB O14920 1/20 0.38
PRKCA P17252 1/20 0.37
PRKCQ Q04759 1/20 0.37
PRKCD Q05655 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5622573 0.95 HTR3A (0.42) CHRNB2CHRNA4PIM1KDM4EMEN1
SCHEMBL5621961 0.87 CHRNB2 (0.43) CHRNB2CHRNA4PIM1GFERHTR3A
SCHEMBL7705451 0.87 CHRNB2 (0.48) CHRNB2CHRNA4PIM1HTR3AHRH4
SCHEMBL5621943 0.85 CHRNB2 (0.44) CHRNB2CHRNA4PIM1HTR3AHRH4
SCHEMBL5620211 0.84 CHRNB2 (0.41) CHRNB2CHRNA4PIM1KDM4EMEN1
SCHEMBL5621910 0.82 HTR3A (0.48) CHRNB2CHRNA4PIM1HTR3APRKCA
SCHEMBL5621369 0.82 CHRM2 (0.41) CHRNB2CHRNA4PIM1GFERHTR3A
SCHEMBL5620167 0.81 PARP1 (0.50) CHRNB2CHRNA4PARP1
SCHEMBL5622576 0.79 ITGB3 (0.42) PIM1KDM4EMEN1KMT2AHTR3A
SCHEMBL5621810 0.77 HTR3A (0.52) KDM4EMEN1KMT2AHTR3ANAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39608-E1 Substituted benzimidazoles and their use as PARP inhibitors ABBOTT GMBH & CO. KG (DE) 2007-05-01 US disclosed
US-6448271-B1 SUCH AS 2-(PIPERIDIN-4-YL)BENZIMIDAZOLE-4-CARBOXAMIDE; INHIBITORS OF ENZYME POLY(ADP-RIBOSE)POLYMERASE; IMPROVED WATER SOLUBILITY BASF AKTIENGESELLSCHAFT (DE) 2002-09-10 US disclosed