SCHEMBL7705471

SCHEMBL7705471

NC(=O)c1cccc2nc(C3CCN(CCc4ccc(O)cc4)C3)[nH]c12

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 14/20 0.62
PARP2 Q9UGN5 2/20 0.48
NR4A2 P43354 1/20 0.40
KCNH2 Q12809 1/20 0.40
LTA4H P09960 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7705626 0.96 PARP1 (0.56) PARP1PARP2NR4A2KCNH2LTA4H
SCHEMBL7706351 0.91 PARP1 (0.61) PARP1PARP2
SCHEMBL7706345 0.91 PARP1 (0.61) PARP1PARP2
SCHEMBL7708486 0.89 PARP1 (0.58) PARP1PARP2KCNH2LTA4H
SCHEMBL5621241 0.89 PARP1 (0.58) PARP1PARP2KCNH2
SCHEMBL7706349 0.89 PARP1 (0.61) PARP1PARP2KCNH2
SCHEMBL7706365 0.88 PARP1 (0.57) PARP1PARP2KCNH2
SCHEMBL5619951 0.87 PARP1 (0.56) PARP1PARP2KCNH2
SCHEMBL7708440 0.87 PARP1 (0.61) PARP1PARP2KCNH2LTA4H
SCHEMBL7706397 0.87 PARP1 (0.55) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448271-B1 SUCH AS 2-(PIPERIDIN-4-YL)BENZIMIDAZOLE-4-CARBOXAMIDE; INHIBITORS OF ENZYME POLY(ADP-RIBOSE)POLYMERASE; IMPROVED WATER SOLUBILITY BASF AKTIENGESELLSCHAFT (DE) 2002-09-10 US disclosed