SCHEMBL7708440

SCHEMBL7708440

NC(=O)c1cccc2nc(C3CCN(CCc4ccc(S(=O)(=O)c5ccccc5)cc4)C3)[nH]c12

nearest known ligand 0.61

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 12/20 0.61
PARP2 Q9UGN5 2/20 0.45
CA12 O43570 5/20 0.41
CA1 P00915 5/20 0.41
CA2 P00918 5/20 0.41
CA4 P22748 5/20 0.41
CA5A P35218 5/20 0.41
CA7 P43166 5/20 0.41
CA9 Q16790 5/20 0.41
CA13 Q8N1Q1 5/20 0.41
CA14 Q9ULX7 5/20 0.41
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
KCNH2 Q12809 1/20 0.40
DRD4 P21917 1/20 0.38
LTA4H P09960 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5621648 0.96 PARP1 (0.56) PARP1PARP2CA12CA1CA2
SCHEMBL7705471 0.87 PARP1 (0.62) PARP1PARP2KCNH2LTA4H
SCHEMBL7706345 0.87 PARP1 (0.61) PARP1PARP2HTR2CDRD4
SCHEMBL7706351 0.87 PARP1 (0.61) PARP1PARP2DRD4
SCHEMBL7708439 0.86 PARP1 (0.83) PARP1PARP2
SCHEMBL7706365 0.85 PARP1 (0.57) PARP1PARP2HTR2AKCNH2
SCHEMBL7708486 0.84 PARP1 (0.58) PARP1PARP2HTR2CKCNH2LTA4H
SCHEMBL5621241 0.84 PARP1 (0.58) PARP1PARP2KCNH2DRD4
SCHEMBL7706349 0.84 PARP1 (0.61) PARP1PARP2KCNH2
SCHEMBL7705626 0.84 PARP1 (0.56) PARP1PARP2KCNH2LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6448271-B1 SUCH AS 2-(PIPERIDIN-4-YL)BENZIMIDAZOLE-4-CARBOXAMIDE; INHIBITORS OF ENZYME POLY(ADP-RIBOSE)POLYMERASE; IMPROVED WATER SOLUBILITY BASF AKTIENGESELLSCHAFT (DE) 2002-09-10 US disclosed