SCHEMBL7705708

SCHEMBL7705708

CS(=O)(=O)c1cccc(C(=O)NCCc2ccccc2)c1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.76
GAA P10253 3/20 0.76
HSD17B10 Q99714 1/20 0.76
RAB9A P51151 8/20 0.75
NPC1 O15118 6/20 0.75
SMN1; SMN2 Q16637 2/20 0.75
TP53 P04637 1/20 0.75
HDAC2 Q92769 2/20 0.64
HDAC8 Q9BY41 2/20 0.64
HDAC6 Q9UBN7 2/20 0.64
HDAC3 O15379 1/20 0.64
HDAC4 P56524 1/20 0.64
HDAC1 Q13547 1/20 0.64
HDAC7 Q8WUI4 1/20 0.64
HDAC10 Q969S8 1/20 0.64
HDAC11 Q96DB2 1/20 0.64
HDAC9 Q9UKV0 1/20 0.64
HDAC5 Q9UQL6 1/20 0.64
HPGD P15428 1/20 0.57
AKR1C3 P42330 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21063806 0.85 RAB9A (0.68) RAB9ANPC1SMN1; SMN2HDAC2HDAC8
SCHEMBL14548357 0.84 RAB9A (0.68) ALDH1A1GAAHSD17B10RAB9ANPC1
SCHEMBL6358306 0.83 ALDH1A1 (0.66) ALDH1A1GAAHSD17B10RAB9ANPC1
SCHEMBL12319476 0.83 ALDH1A1 (0.66) ALDH1A1GAAHSD17B10RAB9ANPC1
SCHEMBL6359372 0.81 SMN1; SMN2 (0.72) ALDH1A1GAAHSD17B10RAB9ANPC1
SCHEMBL18773997 0.80 NPC1 (1.00) ALDH1A1GAARAB9ANPC1SMN1; SMN2
SCHEMBL15676745 0.80 RAB9A (0.74) ALDH1A1RAB9ANPC1SMN1; SMN2TP53
SCHEMBL6842122 0.80 HDAC2 (0.80) ALDH1A1RAB9ANPC1SMN1; SMN2TP53
SCHEMBL13753335 0.80 ALDH1A1 (0.69) ALDH1A1GAAHSD17B10RAB9ANPC1
SCHEMBL19072052 0.80 ALDH1A1 (0.61) ALDH1A1GAAHSD17B10RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901488-B1 2,4-DIAMINOPYRIMIDINE DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2002-11-06 EP disclosed
EP-0901488-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-17 EP disclosed
US-5866583-A Substituted 2,4-diaminopyrimidines HOFFMANN-LA ROCHE INC. (US) 1999-02-02 US disclosed
WO-1997043277-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-11-20 WO disclosed