SCHEMBL12319476

SCHEMBL12319476

CS(=O)(=O)c1cccc(C(=O)NCCO)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.66
HSD17B10 Q99714 2/20 0.66
GAA P10253 2/20 0.66
MEN1 O00255 2/20 0.61
KMT2A Q03164 2/20 0.61
LOX P28300 1/20 0.57
SMN1; SMN2 Q16637 3/20 0.56
RAB9A P51151 2/20 0.52
NPC1 O15118 1/20 0.52
TP53 P04637 1/20 0.52
CYP2C19 P33261 1/20 0.51
NAMPT P43490 1/20 0.50
POLB P06746 1/20 0.49
HPGD P15428 1/20 0.49
HTT P42858 1/20 0.49
CLK2 P49760 1/20 0.48
CDK9 P50750 1/20 0.48
MST1R Q04912 1/20 0.48
CLK4 Q9HAZ1 1/20 0.48
CA12 O43570 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6358306 0.88 ALDH1A1 (0.66) ALDH1A1HSD17B10GAAMEN1KMT2A
SCHEMBL6359372 0.85 SMN1; SMN2 (0.72) ALDH1A1HSD17B10GAAMEN1KMT2A
SCHEMBL13753335 0.84 ALDH1A1 (0.69) ALDH1A1HSD17B10GAAMEN1KMT2A
SCHEMBL19072052 0.84 ALDH1A1 (0.61) ALDH1A1HSD17B10GAAMEN1KMT2A
SCHEMBL12319414 0.84 ALDH1A1 (0.61) ALDH1A1HSD17B10GAAMEN1KMT2A
SCHEMBL7705708 0.83 ALDH1A1 (0.76) ALDH1A1HSD17B10GAAMEN1KMT2A
SCHEMBL14389437 0.82 HSD17B10 (0.60) ALDH1A1HSD17B10GAAMEN1KMT2A
SCHEMBL3319225 0.82 SMN1; SMN2 (0.65) ALDH1A1HSD17B10GAAMEN1KMT2A
SCHEMBL14482756 0.81 ALDH1A1 (0.64) ALDH1A1HSD17B10GAAMEN1KMT2A
SCHEMBL29646375 0.81 ALDH1A1 (0.64) ALDH1A1HSD17B10GAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2114917-B1 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL (JP) 2016-08-10 EP disclosed
US-8933105-B2 Pyrrole compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-01-13 US disclosed
US-8933105-B2 Pyrrole compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-01-13 US disclosed
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed
US-20080262042-A1 1-[5-(2-Fluoropyridin-3-yl)-1-(phenylsulfonyl)-1H-pyrrol-3-yl]-N-methylmethanamine or a salt thereof; acid secretion inhibitor; potassium-competitive acid blocker TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-10-23 US disclosed
US-20080262042-A1 1-[5-(2-Fluoropyridin-3-yl)-1-(phenylsulfonyl)-1H-pyrrol-3-yl]-N-methylmethanamine or a salt thereof; acid secretion inhibitor; potassium-competitive acid blocker TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-10-23 US disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080262042-A1 1-[5-(2-Fluoropyridin-3-yl)-1-(phenylsulfonyl)-1H-pyrrol-3-yl]-N-methylmethanamine or a salt thereof; acid secretion inhibitor; potassium-competitive acid blocker REN, HRH2, ATP4A ALDH1A1 1650/4885HSD17B10 730/4885GAA 549/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.