SCHEMBL7705887

SCHEMBL7705887

O=C(OCC1CC(=O)[C@@H]1COC(=O)c1ccccc1)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.56
PPM1B O75688 1/20 0.49
TDP1 Q9NUW8 2/20 0.49
SLC6A2 P23975 1/20 0.49
SLC6A3 Q01959 1/20 0.49
KMT2A Q03164 1/20 0.49
CHRNB2 P17787 1/20 0.46
CHRNA5 P30532 1/20 0.46
CHRNA7 P36544 1/20 0.46
CHRNA4 P43681 1/20 0.46
FOLH1 Q04609 3/20 0.45
MAPK1 P28482 1/20 0.45
HIF1A Q16665 1/20 0.45
LMNA P02545 2/20 0.44
ALDH1A1 P00352 1/20 0.44
NPC1 O15118 1/20 0.42
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2447972 1.00 CES2 (0.56) CES2PPM1BTDP1SLC6A2SLC6A3
SCHEMBL2447976 1.00 CES2 (0.56) CES2PPM1BTDP1SLC6A2SLC6A3
SCHEMBL2447975 1.00 CES2 (0.56) CES2PPM1BTDP1SLC6A2SLC6A3
SCHEMBL8193371 0.82 CES2 (0.53) CES2PPM1BTDP1SLC6A2SLC6A3
SCHEMBL13286850 0.80 PPM1B (0.56) CES2PPM1BTDP1SLC6A2SLC6A3
SCHEMBL9310364 0.77 TDP1 (0.52) CES2PPM1BTDP1SLC6A2SLC6A3
SCHEMBL3727933 0.76 TDP1 (0.50) CES2PPM1BTDP1SLC6A2SLC6A3
SCHEMBL8191270 0.76 PPM1B (0.52) CES2PPM1BTDP1SLC6A2SLC6A3
SCHEMBL8183690 0.76 PPM1B (0.52) CES2PPM1BTDP1SLC6A2SLC6A3
SCHEMBL7700089 0.75 TDP1 (0.53) TDP1SLC6A2SLC6A3KMT2ACHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6353122-B1 IN CYCLOHEXANONE WITH POTASSIUM PEROXYMONOSULFATE AND SUBSEQUENT REARRANGEMENT TO PROVIDE THE CORRESPONDING CYCLOBUTANONE BRISTOL-MYERS SQUIBB COMPANY 2002-03-05 US disclosed
EP-0433897-B1 Process for preparing an optically active cyclobutane nucleoside SQUIBB & SONS INC (US) 1997-10-01 EP disclosed
EP-0736533-A1 Intermediates and process for the preparation of an antiviral agent BRISTOL-MYERS SQUIBB COMPANY (US) 1996-10-09 EP disclosed
US-5525726-A Process for the preparation of an antiviral agent E. R. SQUIBB & SONS, INC. (US) 1996-06-11 US disclosed
US-5344962-A Intermediates in the synthesis of an optically active cyclobutane nucleoside E. R. SQUIBB & SONS, INC. (US) 1994-09-06 US disclosed
US-5306837-A Intermediates for an optically active cyclobutane nucleoside E. R. SQUIBB & SONS, INC. (US) 1994-04-26 US disclosed
EP-0572209-A2 Process for preparing diprotected 2,3-hydroxymethyl cyclobutanol E.R. SQUIBB & SONS, INC. (US) 1993-12-01 EP disclosed
US-5256806-A Intermediates for the preparation of optically active cyclobutane nucleoside E. R. SQUIBB & SONS, INC. (US) 1993-10-26 US disclosed
US-5237095-A Process for the preparation of an antiviral agent E. R. SQUIBB & SONS, INC. (US) 1993-08-17 US disclosed
US-5233076-A Process for preparing an optically active cyclobutanone, an intermediate in the synthesis of an optically active cyclobutane nucleoside E. R. SQUIBB & SONS, INC. (US) 1993-08-03 US disclosed
US-5218142-A Process for the preparation of an antiviral agent E. R. SQUIBB & SONS, INC. (US) 1993-06-08 US disclosed
US-5198583-A Optically active cyclobutane nucleoside and intermediates, therefor E. R. SQUIBB & SONS, INC. (US) 1993-03-30 US disclosed
US-5185463-A PROCESS FOR THE PREPARATION OF AN ANTIVIRAL AGENT E. R. SQUIBB & SONS, INC. (US) 1993-02-09 US disclosed
US-H1142-H Antiviral agent against herpes and varicella-zoster viruses E. R. SQUIBB & SONS, INC. 1993-02-02 US disclosed
US-5064961-A PROCESS FOR PREPARING AN OPTICALLY ACTIVE CYCLOBUTANE NUCLEOSIDE E. R. SQUIBB & SONS, INC. (US) 1991-11-12 US disclosed
EP-0433897-A2 Process for preparing an optically active cyclobutane nucleoside E.R. SQUIBB & SONS, INC. (US) 1991-06-26 EP disclosed