SCHEMBL7706434

SCHEMBL7706434

CCCOCC1(C)CCCOc2cc(C#Cc3ccc(C(=O)O)cc3)ccc21.CCOCC1(C)CCCOc2cc(C#Cc3ccc(C(=O)O)cc3)ccc21.COCC1(C)CCCOc2cc(C#Cc3ccc(C(=O)O)cc3)ccc21

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
RARB P10826 19/20 0.41
RARG P13631 19/20 0.41
RARA P10276 16/20 0.41
CYP26A1 O43174 1/20 0.41
CYP3A4 P08684 1/20 0.41
CRABP2 P29373 1/20 0.41
RXRA P19793 1/20 0.38
HNF4A P41235 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7137833 0.94 RARB (0.47) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7140796 0.92 RARB (0.48) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7144498 0.90 RARB (0.50) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7140394 0.82 RARB (0.40) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7139553 0.80 RARA (0.47) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7139558 0.80 RARA (0.47) RARBRARGRARACYP26A1CYP3A4
SCHEMBL18247347 0.78 RARB (0.43) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7701222 0.78 RARB (0.45) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7140836 0.77 RARA (0.50) RARBRARGRARACYP26A1CYP3A4
SCHEMBL7140832 0.77 RARA (0.50) RARBRARGRARACYP26A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1212316-A2 BENZOPYRANS AND BENZOTHIOPYRANS AS RAR SELECTIVE RETINOID AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2002-06-12 EP claimed
WO-2001014360-A2 BENZOPYRANS AND BENZOTHIOPYRANS AS RAR SELECTIVE RETINOID AGONISTS F. HOFFMAN-LA ROCHE AG (CH) 2001-03-01 WO claimed