SCHEMBL7706548

SCHEMBL7706548

CCc1nc(-c2ccc(S(C)(=O)=O)cc2)n(-c2ccc(Br)cc2)n1

nearest known ligand 0.56

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.56
ALOX5 P09917 1/20 0.56
PTGS1 P23219 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28181024 0.89 PTGS2 (0.55) PTGS2ALOX5PTGS1
SCHEMBL5203365 0.84 PTGS2 (0.57) PTGS2ALOX5PTGS1
SCHEMBL6885606 0.84 PTGS2 (0.57) PTGS2ALOX5PTGS1
SCHEMBL5202252 0.80 PTGS2 (0.53) PTGS2ALOX5PTGS1
SCHEMBL6880090 0.80 PTGS2 (0.53) PTGS2ALOX5PTGS1
SCHEMBL7706947 0.74 PTGS2 (0.59) PTGS2ALOX5PTGS1
SCHEMBL6884932 0.73 PTGS2 (0.62) PTGS2ALOX5PTGS1
SCHEMBL5205884 0.73 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL6887276 0.72 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL6883989 0.71 PTGS2 (0.64) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1246809-A1 5-ARYL-1H-1,2,4-TRIAZOLE COMPOUNDS AS INHIBITORS OF CYCLOOXYGENASE-2 AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LABORATOIRE THERAMEX (MC) 2002-10-09 EP disclosed
WO-2001034577-A1 5-ARYL-1H-1,2,4-TRIAZOLE COMPOUNDS AS INHIBITORS OF CYCLOOXYGENASE-2 AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LABORATOIRE THERAMEX (MC) 2001-05-17 WO disclosed