SCHEMBL7706815

SCHEMBL7706815

NC(=O)c1ccc(C2=NCCc3ccccc32)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.47
NOS3 P29474 1/20 0.46
NOS2 P35228 1/20 0.46
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
CA7 P43166 2/20 0.44
CA9 Q16790 2/20 0.44
CA14 Q9ULX7 2/20 0.44
MKNK1 Q9BUB5 5/20 0.43
MKNK2 Q9HBH9 4/20 0.43
PLG P00747 1/20 0.43
PLAU P00749 1/20 0.43
PLAT P00750 1/20 0.43
KLK1 P06870 1/20 0.43
MAOA P21397 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
MAPK10 P53779 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21063814 0.87 SRD5A2 (0.50) NOS3NOS2CA1CA2CA7
SCHEMBL7698312 0.82 NOS3 (0.43) NOS3NOS2CA1CA2CA7
SCHEMBL30965936 0.80 CA1 (0.52) NOS3NOS2CA1CA2CA7
SCHEMBL6718892 0.80 NOS3 (0.58) NOS3NOS2CA1CA2CA7
SCHEMBL21063722 0.80 CA1 (0.52) NOS3NOS2CA1CA2CA7
SCHEMBL29384557 0.79 MAPK10 (0.55) NOS3NOS2CA1CA2CA7
SCHEMBL163051 0.79 MAPK10 (0.55) NOS3NOS2CA1CA2CA7
Hydrochloric Acid SCHEMBL27495714 0.77 MAPK10 (0.54) NOS3NOS2CA1CA2CA7
SCHEMBL29498359 0.76 MAPK10 (0.55) NOS3NOS2CA1CA2CA7
SCHEMBL29498358 0.76 MAPK10 (0.55) NOS3NOS2CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1098260-C 2,4-diaminopyrimidine derivatives BASLIR PHARMACEUTICALS AG (CH) 2003-01-08 CN disclosed
EP-0901488-B1 2,4-DIAMINOPYRIMIDINE DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2002-11-06 EP disclosed
CN-1218465-A 2,4-diaminopyrimidine derivatives HOFFMANN LA ROCHE (CH) 1999-06-02 CN disclosed
EP-0901488-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-17 EP disclosed
US-5866583-A Substituted 2,4-diaminopyrimidines HOFFMANN-LA ROCHE INC. (US) 1999-02-02 US disclosed
WO-1997043277-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-11-20 WO disclosed