SCHEMBL7707507

SCHEMBL7707507

CC(C)NC1(C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)CCCC1

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACE P12821 3/20 0.62
ALOX15 P16050 1/20 0.60
ECE1 P42892 10/20 0.58
ITGB2 P05107 2/20 0.57
ICAM1 P05362 2/20 0.57
ITGAL P20701 2/20 0.57
KMT2A Q03164 1/20 0.56
USP2 O75604 1/20 0.55
MAPK1 P28482 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8360275 0.91 ALOX15 (0.61) ACEALOX15ECE1ITGB2ICAM1
SCHEMBL7222010 0.86 ACE (0.63) ACEECE1
SCHEMBL489801 0.84 ECE1 (0.73) ACEALOX15ECE1
SCHEMBL7223833 0.84 ECE1 (0.73) ACEALOX15ECE1
SCHEMBL7230352 0.82 ACE (0.61) ACEALOX15ECE1ITGB2ICAM1
SCHEMBL27798645 0.82 ALOX15 (0.55) ACEALOX15ITGB2ICAM1ITGAL
SCHEMBL19801761 0.80 ACE (0.84) ACEALOX15ECE1
SCHEMBL5193386 0.80 ACE (0.84) ACEALOX15ECE1
SCHEMBL1853071 0.80 ECE1 (0.49) ACEALOX15ECE1ITGB2ICAM1
SCHEMBL15592745 0.78 ACE (0.70) ACEALOX15ECE1ITGB2ICAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6509330-B2 Angiotensin converting enzyme (ACE); neutral endopeptidase (NEP); containing a dipeptide derived from an amino acid, or a conformationally restricted dipeptide mimic BRISTOL-MYERS SQUIBB COMPANY 2003-01-21 US disclosed