SCHEMBL7708028

SCHEMBL7708028

CC1Oc2ccc(C(F)(F)F)cc2N=C1N

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 2/20 0.43
NOS2 P35228 2/20 0.43
NOS1 P29475 1/20 0.43
CTSD P07339 7/20 0.35
BACE1 P56817 1/20 0.34
KIF11 P52732 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
HTR2A P28223 3/20 0.33
HTR2C P28335 3/20 0.33
HTR2B P41595 3/20 0.33
EPHX2 P34913 1/20 0.33
SCN4A P35499 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7988326 0.86 ALDH1A1 (0.35)
SCHEMBL27567477 0.80 NOS3 (0.42) NOS3NOS2NOS1
SCHEMBL6996400 0.79 PIKFYVE (0.32)
Hydrochloric Acid SCHEMBL7711440 0.79 ROCK1 (0.41) NOS3NOS2NOS1HTR2AHTR2C
SCHEMBL7985549 0.76 MAPT (0.43) NOS3NOS2NOS1CTSDHTR2A
SCHEMBL6611984 0.71 PARP1 (0.45) NOS3NOS2NOS1TSHR
SCHEMBL7985616 0.71 MAPT (0.47) NOS3NOS2NOS1HTR2AHTR2C
SCHEMBL7003125 0.71 KCNH2 (0.48)
SCHEMBL5670575 0.70 ESR1 (0.35)
SCHEMBL8119455 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed