SCHEMBL7708086

SCHEMBL7708086

CC1Oc2ccc(C(Cc3ccccc3F)NC(=O)OC(C)(C)C)cc2NC1=O

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
SCN9A Q15858 11/20 0.42
PARP1 P09874 2/20 0.41
IDO1 P14902 1/20 0.39
PTPN1 P18031 1/20 0.39
SMYD3 Q9H7B4 1/20 0.39
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
RCE1 Q9Y256 1/20 0.36
CCKAR P32238 1/20 0.36
CCKBR P32239 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7095873 0.91 CTSS (0.42) CTSSCTSKSCN9AIDO1PTPN1
SCHEMBL7708055 0.90 PARP1 (0.41) SCN9APARP1IDO1SMYD3KDM4E
SCHEMBL7713374 0.88 PARP1 (0.50) CTSSCTSKPARP1IDO1ALDH1A1
SCHEMBL7710779 0.87 TP53 (0.40) PARP1IDO1SMYD3KDM4EALDH1A1
SCHEMBL7704807 0.87 HSD17B10 (0.42) SCN9APARP1IDO1SMYD3
SCHEMBL7708144 0.86 PARP1 (0.42) CTSSCTSKSCN9APARP1IDO1
SCHEMBL7713251 0.85 CTSS (0.45) CTSSCTSKSCN9APARP1IDO1
SCHEMBL7708210 0.84 MC4R (0.41) PARP1IDO1SMYD3KDM4EALDH1A1
SCHEMBL7713294 0.83 PARP1 (0.42) PARP1IDO1SMYD3ALDH1A1CCKAR
SCHEMBL7713338 0.82 PARP1 (0.42) PARP1IDO1SMYD3ALDH1A1CCKAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6365736-B1 TREATMENT OF NERVOUS SYSTEM DISORDERS, CARDIOVASCULAR DISORDERS AND FOR ACTIVITY AS NO-SYNTHASES (NOS) INHIBITORS. SCHERING AKTIENGESELLSCHAFT (DE) 2002-04-02 US disclosed