SCHEMBL7708786

SCHEMBL7708786

Nc1cc(-c2ccccc2F)cc(N)n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.57
FEN1 P39748 4/20 0.49
ALOX5AP P20292 3/20 0.49
MPL P40238 1/20 0.47
MAP4K4 O95819 1/20 0.46
TRPA1 O75762 1/20 0.45
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
ADORA2A P29274 2/20 0.43
NPC1 O15118 2/20 0.43
PTPRC P08575 1/20 0.43
PTPN1 P18031 1/20 0.43
ADORA1 P30542 2/20 0.42
MPO P05164 1/20 0.41
C1R P00736 1/20 0.41
MEN1 O00255 1/20 0.41
PKM P14618 1/20 0.41
NFKB1 P19838 1/20 0.41
MAPK1 P28482 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16506354 0.79 XIAP (0.53) BACE1FEN1ALOX5APMPLMAP4K4
SCHEMBL28116695 0.79 PTPRC (0.54) BACE1FEN1ALOX5APMAP4K4TRPA1
SCHEMBL1337677 0.78 FEN1 (0.47) BACE1FEN1ALOX5APMPLMAP4K4
SCHEMBL7702897 0.75 BACE1 (0.57) BACE1FEN1ALOX5APTRPA1KDM4E
SCHEMBL7709062 0.75 BACE1 (0.57) BACE1FEN1ALOX5APTRPA1KDM4E
SCHEMBL16151213 0.75 ADORA2A (0.49) BACE1MPLMAP4K4TRPA1ADORA2A
SCHEMBL31047274 0.75 ADORA2A (0.49) BACE1MPLMAP4K4TRPA1ADORA2A
SCHEMBL10730124 0.75 ADORA2A (0.49) BACE1TRPA1ADORA2ANPC1PTPRC
SCHEMBL1337206 0.73 BACE1 (0.44) BACE1FEN1ALOX5APMPLMAP4K4
SCHEMBL7711628 0.73 ALOX15 (0.49) KDM4EALDH1A1MEN1NFKB1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed