SCHEMBL7709007

SCHEMBL7709007

Cc1ccc(-c2nc3cc(-c4ccccc4F)cc(N)n3n2)o1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 17/20 0.53
ADORA3 P0DMS8 3/20 0.41
ADORA1 P30542 3/20 0.41
ADORA2B P29275 1/20 0.41
BACE1 P56817 1/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
NFKB1 P19838 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7711726 0.89 ADORA2A (0.54) ADORA2AADORA3ADORA1BACE1NPC1
SCHEMBL7703196 0.87 ADORA2A (0.53) ADORA2AADORA3ADORA1ADORA2BBACE1
SCHEMBL7711762 0.86 ADORA2A (0.52) ADORA2AADORA3ADORA1ADORA2BALDH1A1
SCHEMBL7708964 0.86 ADORA2A (0.52) ADORA2AADORA3ADORA1ADORA2BALDH1A1
SCHEMBL7711685 0.85 ADORA2A (0.57) ADORA2AADORA3ADORA1NPC1ALDH1A1
SCHEMBL7708420 0.85 ADORA2A (0.51) ADORA2AADORA3ADORA1ALDH1A1
SCHEMBL7705853 0.82 ADORA2A (0.53) ADORA2AADORA3ADORA1ADORA2BNPC1
SCHEMBL7487756 0.82 ADORA2A (0.56) ADORA2A
SCHEMBL7708387 0.82 BACE1 (0.40) ADORA2ABACE1NPC1ALDH1A1HPGD
SCHEMBL7711750 0.80 ADORA2A (0.57) ADORA2AADORA3ADORA1NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed