Muscimol

Muscimol

SCHEMBL770913

CCC(=O)O.NCc1cc(O)no1

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 3/20 0.41
CYP2E1 P05181 1/20 0.36
CYP2A6 P11509 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2B6 P20813 1/20 0.36
CYP2C19 P33261 1/20 0.36
PPARA Q07869 1/20 0.36
FFAR3 O14843 1/20 0.34
RAB9A P51151 4/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
NPC1 O15118 3/20 0.33
SMN1; SMN2 Q16637 4/20 0.32
HPGD P15428 2/20 0.32
LMNA P02545 1/20 0.32
S1PR1 P21453 2/20 0.32
S1PR3 Q99500 2/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Muscimol SCHEMBL5781030 0.85 NOTUM (0.47) NOTUMCYP2E1CYP2A6CYP2C9CYP2B6
Muscimol SCHEMBL352714 0.83
Muscimol SCHEMBL8680242 0.83 NOTUM (0.46) NOTUMCYP2E1CYP2A6CYP2C9CYP2B6
Muscimol SCHEMBL7440548 0.83
Hymexazol SCHEMBL7571556 0.77 NPC1 (0.42) CYP2C19FFAR3RAB9AMEN1KMT2A
SCHEMBL7423467 0.76 VHL (0.38) NOTUMPPARAMEN1KMT2ASMN1; SMN2
SCHEMBL8299663 0.73
SCHEMBL595476 0.73 PPARA (0.45) CYP2C19PPARARAB9AMEN1KMT2A
Propionic Acid SCHEMBL22518251 0.72 PPARA (0.36) PPARAFFAR3RAB9AMEN1KMT2A
SCHEMBL9849314 0.72 NOTUM (0.36) NOTUMCYP2E1CYP2A6CYP2C9CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 387 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7053080-B2 Methods and therapeutic combinations for the treatment of obesity using sterol absorption inhibitors SCHERING CORPORATION (US) 2006-05-30 US claimed
CN-111886005-B Use of fluoroethyl normemantine for the prevention and treatment of anxiety 瑞斯特医疗公司 2023-12-15 CN disclosed
US-20220062378-A1 METHODS OF TREATING OR INHIBITING ONSET OF HUNTINGTON'S DISEASE UNIVERSITY OF COPENHAGEN (DK) 2022-03-03 US disclosed
US-20210346469-A1 Compositions and Methods for Increasing Insulin Sensitivity NALPROPION PHARMACEUTICALS LLC (US) 2021-11-11 US disclosed
US-20210198218-A1 COMPOUNDS FOR THERAPEUTIC USE DART NEUROSCIENCE LLC (US) 2021-07-01 US disclosed
EP-3810184-A2 METHODS OF TREATING OR INHIBITING ONSET OF HUNTINGTON'S DISEASE University of Rochester (US) 2021-04-28 EP disclosed
US-10646166-B2 Personal genome information environment providing device, personal genome information environment providing method, and computer program product NATIONAL INSTITUTE OF JAPAN SCIENCE AND TECHNOLOGY AGENCY (JP) 2020-05-12 US disclosed
WO-2020037311-A1 PROTEIN AND PEPTIDE BIOMARKERS FOR TRAUMATIC INJURY TO THE CENTRAL NERVOUS SYSTEM UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2020-02-20 WO disclosed
US-20190290618-A1 Method for Treating Obesity UNIV DUKE (US) 2019-09-26 US disclosed
US-20190262318-A1 Method for Treating Obesity NALPROPION PHARMACEUTICALS LLC 2019-08-29 US disclosed
US-5521297-A Nucleic acids encoding human metabotropic glutamate receptors SALK INSTITUTE BIOTECHNOLOGY/INDUSTRIAL ASSOCIATES (US) 1996-05-28 US disclosed
EP-0701611-A1 HUMAN METABOTROPIC GLUTAMATE RECEPTORS, NUCLEIC ACIDS ENCODING SAME AND USES THEREOF SIBIA NEUROSCIENCES, INC. (US) 1996-03-20 EP disclosed
US-5407935-A 2,3-dihydro-6-nitro-7-sulfamoyl benzo(F)quinoxaline as alpha-amino 3-hydroxy-5-methyl-isoxazole propionic acid antagonist together with probenecid diuretics are useful for treating neurodegenerative diseases WARNER-LAMBERT COMPANY (US) 1995-04-18 US disclosed
WO-1995005600-A1 METHODS OF DETECTING AND COMBATING DISORDERS OF THE CENTRAL NERVOUS SYSTEM DUKE UNIVERSITY (US) 1995-02-23 WO disclosed
WO-1994029449-A1 HUMAN METABOTROPIC GLUTAMATE RECEPTORS, NUCLEIC ACIDS ENCODING SAME AND USES THEREOF THE SALK INSTITUTE BIOTECHNOLOGY/INDUSTRIAL ASSOCIATES, INC. (US) 1994-12-22 WO disclosed
EP-0603301-A1 PHARMACEUTICAL PREPARATION CONTAINING AN URICOSURIC AND AN EXCITATORY AMINO ACID ANTAGONIST WARNER-LAMBERT COMPANY (US) 1994-06-29 EP disclosed
US-5284862-A Neurodegenerative disorders including cerebrovascular disorders; antagonists for excitatory amino acid receptors WARNER-LAMBERT COMPANY (US) 1994-02-08 US disclosed
WO-1993004688-A1 PHARMACEUTICAL PREPARATION CONTAINING AN URICOSURIC AND AN EXCITATORY AMINO ACID ANTAGONIST WARNER-LAMBERT COMPANY (US) 1993-03-18 WO disclosed
WO-1992016205-A2 NOVEL DERIVATIVES OF 2-CARBOXYNDOLES HAVING PHARMACEUTICAL ACTIVITY WARNER-LAMBERT COMPANY (US) 1992-10-01 WO disclosed
US-5145845-A Substituted 2-carboxylindoles having pharmaceutical activity WARNER-LAMBERT CO. (US) 1992-09-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210198218-A1 COMPOUNDS FOR THERAPEUTIC USE OPRK1, ACHE, OPRL1 NOTUM 3998/4885CYP2E1 348/4885CYP2A6 1149/4885
US-20190290618-A1 Method for Treating Obesity SLC6A2, COMT, GAP43 NOTUM 375/4885CYP2E1 150/4885CYP2A6 151/4885
US-20210346469-A1 Compositions and Methods for Increasing Insulin Sensitivity IAPP, GPR119, IRS1 NOTUM 3411/4885CYP2E1 1474/4885CYP2A6 673/4885
US-20190262318-A1 Method for Treating Obesity SLC6A2, COMT, GAP43 NOTUM 375/4885CYP2E1 150/4885CYP2A6 151/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.