SCHEMBL7709150

SCHEMBL7709150

Nc1cccc(-c2cc(N)n3nc(-c4cccs4)nc3c2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.54
ATAD2 Q6PL18 1/20 0.45
DYRK3 O43781 1/20 0.38
CCNT1 O60563 1/20 0.38
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38
CDK9 P50750 1/20 0.38
CDK5 Q00535 1/20 0.38
DYRK1A Q13627 1/20 0.38
CDK5R1 Q15078 1/20 0.38
DYRK2 Q92630 1/20 0.38
DYRK1B Q9Y463 1/20 0.38
FYN P06241 1/20 0.38
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7708740 0.89 ADORA2A (0.57) ADORA2AFYNALDH1A1HPGDL3MBTL1
SCHEMBL7708573 0.88 ADORA2A (0.52) ADORA2AALDH1A1HPGDL3MBTL1MEN1
SCHEMBL7709012 0.85 ADORA2A (0.49) ADORA2ACCNA2CDK2CDK5DYRK1A
SCHEMBL7708503 0.85 NPC1 (0.53) ADORA2ACDK5CDK5R1FYNALDH1A1
SCHEMBL7432234 0.85 ADORA2A (0.56) ADORA2AFYNALDH1A1HPGDL3MBTL1
SCHEMBL7705947 0.83 ADORA2A (0.54) ADORA2AALDH1A1HPGDL3MBTL1MEN1
SCHEMBL7709122 0.82 MAOA (0.47) ADORA2AATAD2ALDH1A1HPGDMEN1
SCHEMBL7705871 0.81 FYN (0.55) ADORA2ADYRK3CCNT1CCNA2CDK2
SCHEMBL7705971 0.80 ADORA2A (0.51) ADORA2AALDH1A1HPGDMEN1KMT2A
SCHEMBL7711729 0.79 ADORA2A (0.52) ADORA2AALDH1A1HPGDL3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed