SCHEMBL7709154

SCHEMBL7709154

Nc1cc(Br)cc2nc(-c3ccco3)nn12.Oc1ccccc1F

nearest known ligand 0.51

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.51
CSNK1A1 P48729 2/20 0.44
CSNK1D P48730 2/20 0.44
CSNK1E P49674 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7427470 0.88 ADORA2A (0.59) ADORA2ACSNK1A1CSNK1DCSNK1E
SCHEMBL7487756 0.78 ADORA2A (0.56) ADORA2A
SCHEMBL7709137 0.77 ADORA2A (0.54) ADORA2A
SCHEMBL7428936 0.75 SMN1; SMN2 (0.44) ADORA2A
SCHEMBL7483266 0.75 ALDH1A1 (0.43) ADORA2A
SCHEMBL7479569 0.73 ADORA2A (0.55) ADORA2A
SCHEMBL7708567 0.73 ADORA2A (0.51) ADORA2ACSNK1A1CSNK1DCSNK1E
SCHEMBL7485299 0.71 ADORA2A (0.56) ADORA2A
SCHEMBL7543025 0.70 ADORA2A (0.41) ADORA2A
SCHEMBL12612295 0.70 ADORA2A (0.68) ADORA2ACSNK1A1CSNK1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed