SCHEMBL7709223

SCHEMBL7709223

N#Cc1ccccc1-c1cc(N)nc(N)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.50
ALOX5AP P20292 1/20 0.49
FEN1 P39748 1/20 0.49
TRPA1 O75762 1/20 0.49
GABRG2 P18507 2/20 0.47
GABRB3 P28472 2/20 0.47
GABRA5 P31644 1/20 0.47
GABRA3 P34903 1/20 0.47
LRRK2 Q5S007 1/20 0.47
ATR Q13535 1/20 0.44
ALDH1A1 P00352 3/20 0.43
KDM4E B2RXH2 1/20 0.43
GAA P10253 1/20 0.43
NR3C1 P04150 1/20 0.41
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
HSD17B10 Q99714 2/20 0.40
GSK3B P49841 1/20 0.40
DYRK1A Q13627 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31663584 0.78 ESR2 (0.50) ESR2TRPA1GABRG2GABRB3GABRA5
SCHEMBL31663620 0.76 GABRG2 (0.67) ESR2TRPA1GABRG2GABRB3GABRA5
SCHEMBL21960122 0.76 ALOX5AP (0.55) ESR2ALOX5APFEN1TRPA1GABRG2
SCHEMBL6169284 0.75 FEN1 (0.57) ESR2ALOX5APFEN1TRPA1GABRG2
SCHEMBL14245039 0.75 ALOX5AP (0.56) ESR2ALOX5APFEN1TRPA1GABRG2
SCHEMBL4359377 0.75 ESR2 (0.66) ESR2ALOX5APFEN1TRPA1GABRG2
SCHEMBL7023813 0.74 ESR2 (0.55) ESR2ALOX5APFEN1TRPA1GABRG2
SCHEMBL979345 0.74 IKBKB (0.50) ESR2ALOX5APFEN1TRPA1GABRG2
SCHEMBL2648336 0.74 ESR2 (0.46) ESR2ALOX5APFEN1TRPA1GABRG2
SCHEMBL223 0.73 ESR2 (0.69) ESR2TRPA1GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6355653-B1 DRUG AND CARRIER FOR ANTIALLERGENS, BRAIN DISORDERS AND NEUROTRANSMITTERS HOFFMANN-LA ROCHE INC. 2002-03-12 US disclosed