SCHEMBL7709266

SCHEMBL7709266

CC(C)(C)[Si](C)(C)OCc1c[nH]c(C(c2ccccc2)(c2ccccc2)c2ccccc2)n1

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.32
TACR1 P25103 1/20 0.31
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6410046 0.76 ALDH1A1 (0.45)
SCHEMBL7802981 0.75 TSHR (0.30)
SCHEMBL6411394 0.75 NOTUM (0.34) MAPK1
SCHEMBL2647015 0.75 DUT (0.31)
Hydrochloric Acid SCHEMBL9670896 0.74
SCHEMBL7832486 0.73 KDM4E (0.41) MAPK1
SCHEMBL6958918 0.73 TDP1 (0.34)
SCHEMBL6457920 0.73 HRH1 (0.37)
SCHEMBL8816412 0.72 NOS2 (0.33)
SCHEMBL9034843 0.72 MEN1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214326-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001017992-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-03-15 WO disclosed
WO-2001018006-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-03-15 WO disclosed
EP-0820445-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1998-01-28 EP disclosed