SCHEMBL7709653

SCHEMBL7709653

CCc1ccc(-c2cccc3c2CCC3=O)c(OCC2(COC(=O)NCc3ccccc3)CC2)c1OC

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.34
GAA P10253 2/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
EPHX1 P07099 2/20 0.33
ATM Q13315 1/20 0.32
TSHR P16473 1/20 0.32
KDM4E B2RXH2 2/20 0.31
HPGD P15428 2/20 0.31
LMNA P02545 1/20 0.31
PKM P14618 1/20 0.31
BCHE P06276 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14737621 0.91 PKM (0.41) ALDH1A1GAAPTGDR2KDM4EHPGD
SCHEMBL7709625 0.85 ALDH1A1 (0.41) ALDH1A1GAAKDM4EHPGD
SCHEMBL7705939 0.82 ALDH1A1 (0.40) ALDH1A1GAAPTGDR2KDM4EHPGD
SCHEMBL14736856 0.82 ALDH1A1 (0.43) ALDH1A1GAAATMKDM4EHPGD
SCHEMBL7716014 0.80 ALDH1A1 (0.36) ALDH1A1GAAKDM4EHPGDLMNA
SCHEMBL7714338 0.77 ALDH1A1 (0.43) ALDH1A1GAATSHRKDM4EHPGD
SCHEMBL14737591 0.77 ALDH1A1 (0.43) ALDH1A1GAATSHRKDM4EHPGD
SCHEMBL2585450 0.76 ALDH1A1 (0.42) ALDH1A1GAAATMTSHRKDM4E
SCHEMBL7712484 0.75 ALDH1A1 (0.33) ALDH1A1GAAKDM4EHPGD
SCHEMBL14737564 0.74 ALDH1A1 (0.42) ALDH1A1GAAKDM4EHPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011134468-A1 BIARYL PHOSPHODIESTERASE INHIBITORS LEO PHARMA A/S (DK) 2011-11-03 WO disclosed