SCHEMBL7709795

SCHEMBL7709795

Nc1c(Br)cc2c3c(cccc13)C(=O)OC2=O

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HKDC1 Q2TB90 1/20 0.65
TYMS P04818 6/20 0.49
CASP6 P55212 1/20 0.39
CTSB P07858 1/20 0.38
TDP1 Q9NUW8 2/20 0.38
ALOX15 P16050 1/20 0.38
MEN1 O00255 2/20 0.37
USP2 O75604 2/20 0.37
KMT2A Q03164 2/20 0.37
RGS12 O14924 1/20 0.37
CYP1A2 P05177 1/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.37
PARP1 P09874 1/20 0.37
MAPT P10636 1/20 0.37
THRB P10828 1/20 0.37
CYP2C9 P11712 1/20 0.37
APEX1 P27695 1/20 0.37
CASP1 P29466 1/20 0.37
BRCA1 P38398 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1133922 0.83 TYMS (0.51) HKDC1TYMSTDP1ALOX15MEN1
SCHEMBL7709652 0.81 TYMS (0.64) HKDC1TYMSTDP1ALOX15MEN1
SCHEMBL10015425 0.79 HKDC1 (1.00) HKDC1CASP6CTSBTDP1MEN1
SCHEMBL11594529 0.79 HKDC1 (0.63) HKDC1CASP6CTSBTDP1MEN1
SCHEMBL10705789 0.79 HKDC1 (0.63) HKDC1TYMSCASP6CTSBTDP1
SCHEMBL29362967 0.77 TYMS (0.61) TYMSMEN1KMT2ACYP1A2POLB
SCHEMBL320954 0.77 TYMS (0.61) TYMSMEN1KMT2ACYP1A2POLB
SCHEMBL7709602 0.76 HKDC1 (0.59) HKDC1TDP1MEN1USP2KMT2A
SCHEMBL11769544 0.75 TYMS (0.44) HKDC1TYMSALOX15CYP1A2CYP3A4
SCHEMBL30608350 0.75 TYMS (0.44) HKDC1TYMSALOX15CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US disclosed
US-6177423-B1 N-(HYDROXY OR PROTECTED HYDROXY)-BENZO(DE)ISOQUINOLINE-1,3-DIONE DERIVATIVES; BACTERIAL DNA GYRASE AND DNA TOPOISOMERASE INHIBITORS USEFUL FOR ANTIBACTERIAL AGENTS HAVING REDUCED DRUG RESISTANCE AND REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed
EP-0939754-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1999-09-08 EP disclosed
WO-1998019648-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed