SCHEMBL7709801

SCHEMBL7709801

O=C1c2cccc3c(/C=N\O)c(CO)cc(c23)C(=O)N1CO

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HEXA P06865 1/20 0.40
HEXB P07686 1/20 0.40
MEN1 O00255 5/20 0.39
KMT2A Q03164 5/20 0.39
MAPT P10636 4/20 0.39
NPC1 O15118 1/20 0.39
AVPR1A P37288 1/20 0.39
RAB9A P51151 1/20 0.39
CLTC Q00610 2/20 0.37
ALDH1A1 P00352 4/20 0.37
USP2 O75604 2/20 0.37
LMNA P02545 2/20 0.37
RGS12 O14924 1/20 0.37
HTT P42858 1/20 0.37
RECQL P46063 1/20 0.37
POLB P06746 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
CYP1B1 Q16678 5/20 0.36
KDM4E B2RXH2 3/20 0.36
KEAP1 Q14145 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7709641 0.73 MAPT (0.48) MEN1KMT2AMAPTNPC1RAB9A
SCHEMBL7709639 0.73 MAPT (0.48) MEN1KMT2AMAPTNPC1RAB9A
SCHEMBL11678307 0.70 HEXA (0.73) HEXAHEXBMEN1KMT2AMAPT
SCHEMBL6311388 0.66 MEN1 (0.81) MEN1KMT2AMAPTNPC1AVPR1A
SCHEMBL101555 0.64 CA12 (0.59) MEN1KMT2AMAPTRAB9AALDH1A1
SCHEMBL30523037 0.64 CA12 (0.59) MEN1KMT2AMAPTRAB9AALDH1A1
SCHEMBL13496074 0.62 KMT2A (0.42) MEN1KMT2AMAPTCLTCALDH1A1
Fluoride SCHEMBL28030878 0.62 CA12 (0.57) MEN1KMT2AMAPTRAB9AALDH1A1
SCHEMBL23843535 0.62 MEN1 (0.47) HEXAHEXBMEN1KMT2AMAPT
SCHEMBL19770240 0.61 TERT (0.60) HEXAHEXBMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US claimed
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US disclosed
US-6177423-B1 N-(HYDROXY OR PROTECTED HYDROXY)-BENZO(DE)ISOQUINOLINE-1,3-DIONE DERIVATIVES; BACTERIAL DNA GYRASE AND DNA TOPOISOMERASE INHIBITORS USEFUL FOR ANTIBACTERIAL AGENTS HAVING REDUCED DRUG RESISTANCE AND REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed