SCHEMBL7712151

SCHEMBL7712151

Nc1cc2c3c(ccc([N+](=O)[O-])c3c1[N+](=O)[O-])C(=O)OC2=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.46
ACHE P22303 1/20 0.46
CES1 P23141 1/20 0.46
ALDH1A1 P00352 2/20 0.43
TDP1 Q9NUW8 4/20 0.39
TSHR P16473 2/20 0.39
MAPT P10636 2/20 0.37
MCL1 Q07820 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
POLB P06746 1/20 0.36
CYP3A4 P08684 1/20 0.36
ALOX15 P16050 1/20 0.36
TYMS P04818 4/20 0.35
LMNA P02545 1/20 0.35
HSP90AA1 P07900 1/20 0.35
CDK5 Q00535 1/20 0.35
CDK5R1 Q15078 1/20 0.35
MAPK1 P28482 1/20 0.35
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7709784 0.86 BCHE (0.46) BCHEACHECES1ALDH1A1TDP1
SCHEMBL7703711 0.83 BCHE (0.46) BCHEACHECES1ALDH1A1MAPT
SCHEMBL4150369 0.81 BCHE (0.68) BCHEACHECES1ALDH1A1TDP1
SCHEMBL7709620 0.80 LMNA (0.44) BCHEACHECES1ALDH1A1TDP1
SCHEMBL7703712 0.78 TYMS (0.44) ALDH1A1TDP1MAPTMEN1KMT2A
SCHEMBL7709651 0.75 BCHE (0.47) BCHEACHECES1ALDH1A1TDP1
SCHEMBL27874944 0.75 BCHE (0.59) BCHEACHECES1ALDH1A1TDP1
SCHEMBL30659874 0.72 ALDH1A1 (0.47) ALDH1A1TDP1TSHRMAPTMCL1
SCHEMBL10941035 0.72 ALDH1A1 (0.47) ALDH1A1TDP1TSHRMAPTMCL1
SCHEMBL5142990 0.71 ALDH1A1 (0.57) BCHEACHECES1ALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US disclosed
US-6177423-B1 N-(HYDROXY OR PROTECTED HYDROXY)-BENZO(DE)ISOQUINOLINE-1,3-DIONE DERIVATIVES; BACTERIAL DNA GYRASE AND DNA TOPOISOMERASE INHIBITORS USEFUL FOR ANTIBACTERIAL AGENTS HAVING REDUCED DRUG RESISTANCE AND REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed
EP-0939754-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1999-09-08 EP disclosed
WO-1998019648-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed