SCHEMBL7703712

SCHEMBL7703712

Nc1cc2c3c(cccc3c1[N+](=O)[O-])C(=O)OC2=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 10/20 0.44
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
MAPT P10636 2/20 0.40
LMNA P02545 1/20 0.39
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
CYP3A4 P08684 2/20 0.37
USP2 O75604 2/20 0.36
RGS12 O14924 1/20 0.36
CYP1A2 P05177 1/20 0.36
POLB P06746 1/20 0.36
PARP1 P09874 1/20 0.36
THRB P10828 1/20 0.36
CYP2C9 P11712 1/20 0.36
APEX1 P27695 1/20 0.36
CASP1 P29466 1/20 0.36
BRCA1 P38398 1/20 0.36
MTOR P42345 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1133994 0.82 TYMS (0.44) TYMSALDH1A1MEN1KMT2AMAPT
SCHEMBL7709458 0.82 MEN1 (0.57) TYMSALDH1A1MEN1KMT2AMAPT
SCHEMBL7712218 0.79 KMT2A (0.46) TYMSALDH1A1MEN1KMT2AMAPT
SCHEMBL7712151 0.78 BCHE (0.46) TYMSALDH1A1MEN1KMT2AMAPT
SCHEMBL1133922 0.78 TYMS (0.51) TYMSALDH1A1MEN1KMT2AMAPT
SCHEMBL7709571 0.75 TYMS (0.57) TYMSALDH1A1MEN1KMT2AMAPT
SCHEMBL4077252 0.75 TYMS (0.49) TYMSALDH1A1MEN1KMT2AMAPT
SCHEMBL29836499 0.75 TYMS (0.49) TYMSALDH1A1MEN1KMT2AMAPT
SCHEMBL29665023 0.73 TYMS (0.44) TYMSALDH1A1MEN1KMT2ALMNA
SCHEMBL4084412 0.73 TYMS (0.44) TYMSALDH1A1MEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362181-B1 BACTERICIDES; ENZYME INHIBITORS; ANTITUMOR AGENTS WARNER-LAMBERT COMPANY 2002-03-26 US disclosed
US-6177423-B1 N-(HYDROXY OR PROTECTED HYDROXY)-BENZO(DE)ISOQUINOLINE-1,3-DIONE DERIVATIVES; BACTERIAL DNA GYRASE AND DNA TOPOISOMERASE INHIBITORS USEFUL FOR ANTIBACTERIAL AGENTS HAVING REDUCED DRUG RESISTANCE AND REDUCED SIDE EFFECTS WARNER-LAMBERT COMPANY 2001-01-23 US disclosed
EP-0939754-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1999-09-08 EP disclosed
WO-1998019648-A2 N-OXY-NAPHTHALIMIDES AS ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY (US) 1998-05-14 WO disclosed