SCHEMBL7715665

SCHEMBL7715665

CCc1ccc(-c2cccc3c2CCC3=O)c(OCC(C)(C)C(=O)NC)c1OC

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
GAA P10253 1/20 0.38
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
SSTR4 P31391 5/20 0.32
SSTR1 P30872 1/20 0.32
ADRB2 P07550 1/20 0.32
ADRB1 P08588 1/20 0.32
HTR1A P08908 1/20 0.32
ADRB3 P13945 1/20 0.32
TSHR P16473 1/20 0.32
SLC6A4 P31645 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
BRAF P15056 1/20 0.31
S1PR1 P21453 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2585854 0.89 ALDH1A1 (0.48) ALDH1A1GAAKDM4EHPGDSSTR4
SCHEMBL7717394 0.89 ALDH1A1 (0.39) ALDH1A1GAAKDM4EHPGDADRB2
SCHEMBL7712445 0.87 ALDH1A1 (0.38) ALDH1A1GAAKDM4EHPGDADRB2
SCHEMBL7713141 0.84 ALDH1A1 (0.40) ALDH1A1GAAKDM4EHPGDADRB2
SCHEMBL7714650 0.83 ALDH1A1 (0.40) ALDH1A1GAAKDM4EHPGDADRB2
SCHEMBL2591327 0.82 ALDH1A1 (0.46) ALDH1A1GAAKDM4EHPGDSSTR4
SCHEMBL2588129 0.79 ALDH1A1 (0.50) ALDH1A1GAAKDM4EHPGDADRB2
SCHEMBL2591184 0.78 KDM4E (0.45) ALDH1A1KDM4EHPGDSSTR4SSTR1
SCHEMBL2591573 0.78 ALDH1A1 (0.51) ALDH1A1GAAKDM4EHPGDADRB2
SCHEMBL2592229 0.77 ALDH1A1 (0.48) ALDH1A1GAAKDM4EHPGDADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011134468-A1 BIARYL PHOSPHODIESTERASE INHIBITORS LEO PHARMA A/S (DK) 2011-11-03 WO disclosed