SCHEMBL7716641

SCHEMBL7716641

CC(C)N(C=Nc1ncc(Oc2ccc(Cl)cc2)c(N2CCN(CCO)CC2)n1)C(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.37
METAP1 P53582 1/20 0.36
HRH4 Q9H3N8 1/20 0.36
ROCK2 O75116 3/20 0.35
ROCK1 Q13464 3/20 0.35
HPGD P15428 4/20 0.35
HTT P42858 4/20 0.35
MAPT P10636 3/20 0.35
TSHR P16473 2/20 0.35
RAB9A P51151 2/20 0.35
KDM4E B2RXH2 2/20 0.35
RXFP1 Q9HBX9 1/20 0.34
ALDH1A1 P00352 2/20 0.34
HSD17B10 Q99714 1/20 0.34
LRRK2 Q5S007 1/20 0.34
MDM2 Q00987 1/20 0.33
CFTR P13569 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
KMT2A Q03164 1/20 0.33
MAPK14 Q16539 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7716638 1.00 LMNA (0.37) LMNAMETAP1HRH4ROCK2ROCK1
SCHEMBL8138459 0.90 KDM4E (0.33) LMNAMETAP1HRH4HPGDHTT
SCHEMBL7714501 0.79 LMNA (0.46) LMNAMETAP1HRH4ROCK2ROCK1
SCHEMBL7716737 0.78 ALDH1A1 (0.48) LMNAMETAP1HRH4HPGDHTT
SCHEMBL7714319 0.78 LMNA (0.41) LMNAMETAP1HRH4ROCK2ROCK1
SCHEMBL7714708 0.78 LMNA (0.46) LMNAMETAP1HRH4ROCK2ROCK1
SCHEMBL7708442 0.77 LMNA (0.45) LMNAMETAP1HRH4ROCK2ROCK1
SCHEMBL5202933 0.77 L3MBTL1 (0.35) HTTMAPTKDM4EALDH1A1KMT2A
SCHEMBL5202927 0.77 L3MBTL1 (0.35) HTTMAPTKDM4EALDH1A1KMT2A
SCHEMBL7714147 0.76 ALDH1A1 (0.44) LMNAMETAP1HRH4HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6440965-B1 Substituted pyrimidine derivatives, their preparation and their use in the treatment of neurodegenerative or neurological disorders of the central nervous system KRENITSKY PHARMACEUTICALS, INC. 2002-08-27 US disclosed