SCHEMBL7716899

SCHEMBL7716899

COC(=O)Cc1ccc(NCC(C)N(CC(O[Si](C)(C)C(C)(C)C)c2cccc(Cl)c2)C(=O)OC(C)(C)C)c(C)c1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 3/20 0.33
ADRB3 P13945 3/20 0.33
ADRB1 P08588 2/20 0.33
GLA P06280 1/20 0.33
RPS6KB1 P23443 1/20 0.30
IGF1R P08069 1/20 0.30
CYP3A4 P08684 1/20 0.30
ITGB1 P05556 1/20 0.30
ITGA4 P13612 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7708894 0.92 ADRB2 (0.32) ADRB2ADRB3ADRB1GLARPS6KB1
SCHEMBL7714622 0.88
SCHEMBL7712721 0.86 RPS6KB1 (0.30) RPS6KB1
SCHEMBL7716950 0.85 ADRB2 (0.32) ADRB2ADRB3ADRB1ITGB1ITGA4
SCHEMBL7714945 0.84 CYP3A4 (0.30) CYP3A4
SCHEMBL7714803 0.84 PDCD1 (0.33)
SCHEMBL7714670 0.84 ADRB2 (0.33) ADRB2ADRB3ADRB1GLAITGB1
SCHEMBL7714532 0.82 ADRB2 (0.32) ADRB2ADRB3ADRB1CYP3A4
SCHEMBL7709011 0.81 NR1H2 (0.32) ADRB2ADRB3ADRB1ITGB1ITGA4
SCHEMBL7712843 0.80 CTSS (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865421-B1 ARYLETHANOLAMINE DERIVATIVES AND THEIR USE AS AGONISTS OF ATYPICAL BETA-ADRENOCEPTORS GLAXO GROUP LTD (GB) 2002-03-27 EP disclosed
US-6048872-A DIETETICS; ANTIDIABETIC AGENTS; CARDIOVASCULAR DISORDERS; GASTROINTESTINAL DISORDERS GLAXO WELLCOME INC. (US) 2000-04-11 US disclosed