SCHEMBL7717535

SCHEMBL7717535

COC(=O)c1ccc(C#CC(=O)c2ccc3c(c2)C(C)(C)CCC3(C)C)cc1O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.52
RARB P10826 6/20 0.49
CYP26A1 O43174 5/20 0.49
RARG P13631 5/20 0.49
RARA P10276 4/20 0.49
CRABP2 P29373 1/20 0.49
CYP26B1 Q9NR63 1/20 0.43
RXRA P19793 8/20 0.41
RXRB P28702 5/20 0.41
RXRG P48443 4/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
PDK2 Q15119 1/20 0.40
PDK4 Q16654 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7714910 0.88 RARB (0.58) CYP3A4RARBCYP26A1RARGRARA
SCHEMBL7937802 0.88 RXRA (0.41) CYP3A4RARBCYP26A1RARGRARA
SCHEMBL19342969 0.87 RARB (0.56) CYP3A4RARBCYP26A1RARGRARA
SCHEMBL7928392 0.87 RXRA (0.40) CYP3A4RARBCYP26A1RARGRARA
SCHEMBL7709220 0.86 CYP3A4 (0.65) CYP3A4RARBCYP26A1RARGRARA
SCHEMBL7714846 0.86 RARA (0.52) CYP3A4RARBCYP26A1RARGRARA
SCHEMBL7752278 0.80 CYP3A4 (0.44) CYP3A4RARBCYP26A1RARGRARA
SCHEMBL6876627 0.80 CYP3A4 (0.43) CYP3A4RARBCYP26A1RARGRARA
SCHEMBL7714935 0.79 RARB (0.42) CYP3A4RARBCYP26A1RARGRARA
SCHEMBL7713094 0.78 CYP3A4 (0.41) CYP3A4RARBCYP26A1RARGRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6368608-B1 SKIN DISORDERS CENTRE INTERNATIONAL DE RECHERCHE DERMATOLOGIQUES GALDERMA (C.I.R.D.) (FR) 2002-04-09 US disclosed
US-6162445-A Polyaromatic propynyl compounds and pharmaceutical/cosmetic compositions comprised thereof CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (FR) 2000-12-19 US disclosed