SCHEMBL7714846

SCHEMBL7714846

COC(=O)c1ccc(C#CC(=O)c2ccc3c(c2)C(C)(C)CCS3)cc1O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 10/20 0.52
RARB P10826 10/20 0.52
RARG P13631 10/20 0.52
CYP3A4 P08684 4/20 0.49
KMT2A Q03164 1/20 0.49
CYP26A1 O43174 2/20 0.48
RXRA P19793 2/20 0.40
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
ALOX15 P16050 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
PDK2 Q15119 1/20 0.36
PDK4 Q16654 1/20 0.36
CA9 Q16790 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7713111 0.89 CYP3A4 (0.55) RARARARBRARGCYP3A4KMT2A
SCHEMBL8440028 0.89 RARA (0.54) RARARARBRARGCYP3A4KMT2A
SCHEMBL7717535 0.86 CYP3A4 (0.52) RARARARBRARGCYP3A4KMT2A
SCHEMBL7937802 0.82 RXRA (0.41) RARARARBRARGCYP3A4CYP26A1
SCHEMBL7713085 0.81 RARA (0.45) RARARARBRARGCYP3A4KMT2A
SCHEMBL7928392 0.80 RXRA (0.40) RARARARBRARGCYP3A4CYP26A1
SCHEMBL19342893 0.79 RARA (0.65) RARARARBRARGCYP3A4KMT2A
SCHEMBL9256097 0.79 CYP3A4 (0.57) RARARARBRARGCYP3A4KMT2A
SCHEMBL19342892 0.79 RARB (0.54) RARARARBRARGCYP3A4KMT2A
SCHEMBL19342908 0.78 RARA (0.53) RARARARBRARGCYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6368608-B1 SKIN DISORDERS CENTRE INTERNATIONAL DE RECHERCHE DERMATOLOGIQUES GALDERMA (C.I.R.D.) (FR) 2002-04-09 US disclosed
US-6162445-A Polyaromatic propynyl compounds and pharmaceutical/cosmetic compositions comprised thereof CENTRE INTERNATIONAL DE RECHERCHES DERMATOLOGIQUES GALDERMA (FR) 2000-12-19 US disclosed