SCHEMBL7717581

SCHEMBL7717581

CC(C)(C)OC(=O)Nc1c([Si](C)(C)C)ccc2ccc(CS(=O)(=O)O)cc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.40
TOP2A P11388 1/20 0.37
TOP2B Q02880 1/20 0.37
CYP17A1 P05093 1/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
RAB9A P51151 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA7 P43166 1/20 0.36
CA14 Q9ULX7 1/20 0.36
MAPK14 Q16539 1/20 0.35
LCK P06239 4/20 0.35
P2RX3 P56373 1/20 0.35
SCN9A Q15858 1/20 0.34
NPSR1 Q6W5P4 4/20 0.34
JAK2 O60674 3/20 0.34
HPGD P15428 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7715090 0.81 NQO2 (0.49) NQO2TOP2ATOP2BKMT2AMEN1
SCHEMBL7719307 0.80 NQO2 (0.46) NQO2CA12CA1CA7CA14
SCHEMBL7717601 0.79 ALDH1A1 (0.37) NQO2TOP2ATOP2BKMT2AMEN1
SCHEMBL7717631 0.74 GAA (0.36) NQO2TOP2ATOP2BKMT2AMEN1
SCHEMBL7719470 0.71 KCNQ4 (0.39) CYP17A1KMT2ACA12CA1CA7
SCHEMBL27351496 0.67 LCK (0.52) KMT2AMEN1NPC1GAARAB9A
SCHEMBL7717690 0.64 NQO2 (0.51) NQO2TOP2ATOP2BKMT2AMEN1
SCHEMBL24150453 0.63 NQO2 (0.42) NQO2KMT2AMEN1NPC1GAA
SCHEMBL24150706 0.63 LCK (0.45) NQO2NPC1RAB9ACA12CA1
SCHEMBL23028526 0.63 BRD4 (0.46) NQO2CYP17A1NPSR1ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441017-B1 Inhibitors of prenyl-protein transferase MERCK & CO., INC. 2002-08-27 US disclosed