SCHEMBL7717601

SCHEMBL7717601

CC(C)(C)OC(=O)Nc1c([Si](C)(C)C)ccc2ccc(OS(C)(=O)=O)cc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
NQO2 P16083 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ATR Q13535 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KAT6A Q92794 1/20 0.34
GAA P10253 4/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA9 Q16790 1/20 0.33
LCK P06239 3/20 0.33
IDH1 O75874 1/20 0.33
HPGD P15428 3/20 0.33
KDM4E B2RXH2 3/20 0.33
GLA P06280 2/20 0.33
MAPT P10636 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7709280 0.84 ALDH1A1 (0.39) ALDH1A1NQO2NPSR1ATRSMN1; SMN2
SCHEMBL7715090 0.82 NQO2 (0.49) NQO2NPSR1ATRGAAMEN1
SCHEMBL7717631 0.81 GAA (0.36) ALDH1A1NQO2NPSR1ATRGAA
SCHEMBL7717581 0.79 NQO2 (0.40) ALDH1A1NQO2NPSR1ATRKAT6A
SCHEMBL487112 0.78 TRPV1 (0.44) ALDH1A1NQO2KAT6AMEN1NPC1
SCHEMBL1530133 0.71 ENPP3 (0.52) ALDH1A1MEN1KMT2ACA12CA1
SCHEMBL7714920 0.71 MEN1 (0.42) NQO2NPSR1KAT6AGAAMEN1
SCHEMBL10062583 0.70 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2KAT6AGAACA12
SCHEMBL486679 0.70 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2GAACA12CA1
SCHEMBL7714050 0.70 CA12 (0.41) ALDH1A1NQO2NPSR1ATRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441017-B1 Inhibitors of prenyl-protein transferase MERCK & CO., INC. 2002-08-27 US disclosed
EP-1214326-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 2002-06-19 EP disclosed
WO-2001018006-A1 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2001-03-15 WO disclosed